METHODS FOR PRODUCING ANGIOTENSINE II ANTAGONISTIC BENZIMIDAZOLE AND INDOLE DERIVATIVES AND MEDICAL PREPARATIVES CONTAINING THEM

This invention provides pharmaceutical heterocyclic derivatives of the formula in which R3 are specified nitrogen-containing fused rings. They antagonize angiotensin II receptors in mammals.

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Hauptverfasser: THRASHER,KENNETH JEFF,US, BOYD,DONALD BRADFORD,US, REEL,JON KEVIN,US, VASUDEVAN,VENKATRAGHAVAN,US, WHITESITT,CELIA ANN,US, PALKOWITZ,ALAN DAVID,US, SIMON,RICHARD LEE,US, LIFER,SHERRYL LYNN,US, PFEIFER,WILLIAM,US, STEINBERG,MITCHELL IRWIN,US, MARSHALL,WINSTON STANLEY,US
Format: Patent
Sprache:eng
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Zusammenfassung:This invention provides pharmaceutical heterocyclic derivatives of the formula in which R3 are specified nitrogen-containing fused rings. They antagonize angiotensin II receptors in mammals.