NOVEL COMPOUNDS
Spoj formule (I) naznačen time da, R1 i R3 je isti ili različit, te je nezavisno odabran od H, (C1-C6) alkil, (C3-C7) cikloalkil, halo, CN, OF3, -O-(C1-C6)alkil, -CO2-(C1-C6)alkil, COOH, -CONH-(C1-C6)alkil, -CONH-aril, -NH2, -CONH-R6, The present invention discloses a novel thyroid like compounds of...
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| creator | SHITALKUMAR PUKHARAJ ZAMBAD ASHOK KASUNDRA RAMESH GUPTA M. AMIR SIDDIQUI LAXMIKANT CHHIPA DAVINDER TULI VIJAY CHAUTHAIWALE C. DUTT SIRALEE MUNSHI SUBRAT KUMAR BHATTAMISRA |
| description | Spoj formule (I) naznačen time da, R1 i R3 je isti ili različit, te je nezavisno odabran od H, (C1-C6) alkil, (C3-C7) cikloalkil, halo, CN, OF3, -O-(C1-C6)alkil, -CO2-(C1-C6)alkil, COOH, -CONH-(C1-C6)alkil, -CONH-aril, -NH2, -CONH-R6,
The present invention discloses a novel thyroid like compounds of formula (I), wherein R1 R2, R3, R4 and Z are as defined in the specification, method for its preparation, composition containing such compounds and use of such compounds and composition as medicament. Further, compounds of formula (I) has significantly low binding affinity to thyroid receptors and thus considerably devoid of thyrotoxic effects. The invention also relates to the use of the compound of formula (I) for the preparation of a medicament for treating various disease conditions such as obesity, dyslipidemia, metabolic syndrome and co-morbidities associated with metabolic syndrome. |
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The present invention discloses a novel thyroid like compounds of formula (I), wherein R1 R2, R3, R4 and Z are as defined in the specification, method for its preparation, composition containing such compounds and use of such compounds and composition as medicament. Further, compounds of formula (I) has significantly low binding affinity to thyroid receptors and thus considerably devoid of thyrotoxic effects. The invention also relates to the use of the compound of formula (I) for the preparation of a medicament for treating various disease conditions such as obesity, dyslipidemia, metabolic syndrome and co-morbidities associated with metabolic syndrome.</description><language>hrv ; eng</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2010</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20101231&DB=EPODOC&CC=HR&NR=P20100611T1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20101231&DB=EPODOC&CC=HR&NR=P20100611T1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>SHITALKUMAR PUKHARAJ ZAMBAD</creatorcontrib><creatorcontrib>ASHOK KASUNDRA</creatorcontrib><creatorcontrib>RAMESH GUPTA</creatorcontrib><creatorcontrib>M. AMIR SIDDIQUI</creatorcontrib><creatorcontrib>LAXMIKANT CHHIPA</creatorcontrib><creatorcontrib>DAVINDER TULI</creatorcontrib><creatorcontrib>VIJAY CHAUTHAIWALE</creatorcontrib><creatorcontrib>C. DUTT</creatorcontrib><creatorcontrib>SIRALEE MUNSHI</creatorcontrib><creatorcontrib>SUBRAT KUMAR BHATTAMISRA</creatorcontrib><title>NOVEL COMPOUNDS</title><description>Spoj formule (I) naznačen time da, R1 i R3 je isti ili različit, te je nezavisno odabran od H, (C1-C6) alkil, (C3-C7) cikloalkil, halo, CN, OF3, -O-(C1-C6)alkil, -CO2-(C1-C6)alkil, COOH, -CONH-(C1-C6)alkil, -CONH-aril, -NH2, -CONH-R6,
The present invention discloses a novel thyroid like compounds of formula (I), wherein R1 R2, R3, R4 and Z are as defined in the specification, method for its preparation, composition containing such compounds and use of such compounds and composition as medicament. Further, compounds of formula (I) has significantly low binding affinity to thyroid receptors and thus considerably devoid of thyrotoxic effects. The invention also relates to the use of the compound of formula (I) for the preparation of a medicament for treating various disease conditions such as obesity, dyslipidemia, metabolic syndrome and co-morbidities associated with metabolic syndrome.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2010</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZOD38w9z9VFw9vcN8A_1cwnmYWBNS8wpTuWF0twMym6uIc4euqkF-fGpxQWJyal5qSXxHkEBRgaGBgZmhoYhIYbGxKkCAG_kHq4</recordid><startdate>20101231</startdate><enddate>20101231</enddate><creator>SHITALKUMAR PUKHARAJ ZAMBAD</creator><creator>ASHOK KASUNDRA</creator><creator>RAMESH GUPTA</creator><creator>M. AMIR SIDDIQUI</creator><creator>LAXMIKANT CHHIPA</creator><creator>DAVINDER TULI</creator><creator>VIJAY CHAUTHAIWALE</creator><creator>C. DUTT</creator><creator>SIRALEE MUNSHI</creator><creator>SUBRAT KUMAR BHATTAMISRA</creator><scope>EVB</scope></search><sort><creationdate>20101231</creationdate><title>NOVEL COMPOUNDS</title><author>SHITALKUMAR PUKHARAJ ZAMBAD ; ASHOK KASUNDRA ; RAMESH GUPTA ; M. AMIR SIDDIQUI ; LAXMIKANT CHHIPA ; DAVINDER TULI ; VIJAY CHAUTHAIWALE ; C. DUTT ; SIRALEE MUNSHI ; SUBRAT KUMAR BHATTAMISRA</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_HRP20100611TT13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>hrv ; eng</language><creationdate>2010</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>SHITALKUMAR PUKHARAJ ZAMBAD</creatorcontrib><creatorcontrib>ASHOK KASUNDRA</creatorcontrib><creatorcontrib>RAMESH GUPTA</creatorcontrib><creatorcontrib>M. AMIR SIDDIQUI</creatorcontrib><creatorcontrib>LAXMIKANT CHHIPA</creatorcontrib><creatorcontrib>DAVINDER TULI</creatorcontrib><creatorcontrib>VIJAY CHAUTHAIWALE</creatorcontrib><creatorcontrib>C. DUTT</creatorcontrib><creatorcontrib>SIRALEE MUNSHI</creatorcontrib><creatorcontrib>SUBRAT KUMAR BHATTAMISRA</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>SHITALKUMAR PUKHARAJ ZAMBAD</au><au>ASHOK KASUNDRA</au><au>RAMESH GUPTA</au><au>M. AMIR SIDDIQUI</au><au>LAXMIKANT CHHIPA</au><au>DAVINDER TULI</au><au>VIJAY CHAUTHAIWALE</au><au>C. DUTT</au><au>SIRALEE MUNSHI</au><au>SUBRAT KUMAR BHATTAMISRA</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>NOVEL COMPOUNDS</title><date>2010-12-31</date><risdate>2010</risdate><abstract>Spoj formule (I) naznačen time da, R1 i R3 je isti ili različit, te je nezavisno odabran od H, (C1-C6) alkil, (C3-C7) cikloalkil, halo, CN, OF3, -O-(C1-C6)alkil, -CO2-(C1-C6)alkil, COOH, -CONH-(C1-C6)alkil, -CONH-aril, -NH2, -CONH-R6,
The present invention discloses a novel thyroid like compounds of formula (I), wherein R1 R2, R3, R4 and Z are as defined in the specification, method for its preparation, composition containing such compounds and use of such compounds and composition as medicament. Further, compounds of formula (I) has significantly low binding affinity to thyroid receptors and thus considerably devoid of thyrotoxic effects. The invention also relates to the use of the compound of formula (I) for the preparation of a medicament for treating various disease conditions such as obesity, dyslipidemia, metabolic syndrome and co-morbidities associated with metabolic syndrome.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | NOVEL COMPOUNDS |
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