Derivados de acetamida N-piperidinilo como bloqueadores de canales de calcio

Derivados de acetamida N-piperidinilo como bloqueadores de canales de calcio

Un compuesto con la estructura: **Fórmula** o una sal farmacéuticamente aceptable de los mismos, para uso en el tratamiento del dolor crónico o agudo. Methods and compounds effective in ameliorating conditions characterized by unwanted calcium channel activity, particularly unwanted T-type calcium c...

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Bibliographische Detailangaben
Hauptverfasser: PAJOUHESH, Hassan, TAN, Jason, CHAKKA, Nagasree, KAUL, Ramesh, ZHU, Yongbao, ZHOU, Yuanxi, DING, Yanbing, GRIMWOOD, Mike, ZHANG, Lingyun
Format: Patent
Sprache:spa
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Zusammenfassung:Un compuesto con la estructura: **Fórmula** o una sal farmacéuticamente aceptable de los mismos, para uso en el tratamiento del dolor crónico o agudo. Methods and compounds effective in ameliorating conditions characterized by unwanted calcium channel activity, particularly unwanted T-type calcium channel activity, are disclosed. Specifically, a series of compounds which are N-piperidinyl acetamide derivatives as shown in formula (1) are disclosed as calcium ion channel activating modulators. Compositions comprising these compounds and the use of these compounds in the treatment or prevention of conditions such as epilepsy are also disclosed.