PIRAZOLILO TRIDENTADO BIFUNCIONAL QUE CONTIENE LIGANDOS PARA COMPLEJOS DE TRICARBONILO RE, TC Y MN
Agente quelante de la fórmula general: **(Ver fórmula)** en la que m es 0 ó 1 X es NR4; Y es NHR5, SR5 o P(R5)2; R1 y R3 son iguales o diferentes y se seleccionan entre H, alquilo o arilo; R2 es H, COOH, NHR6 o (CH2)nCOOR6; R4 es (CH2)nCOOR6, o (CH2)nOR6; R5 es H, alquilo, arilo, (CH2) nCOOR6, o (CH...
Gespeichert in:
| Hauptverfasser: | , , , , |
|---|---|
| Format: | Patent |
| Sprache: | spa |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | ROCHA PAULO, ANTONIO, M GALAMBA CORREIA, JOAO, D ALVES, SUSANA VITOR, RUTE SANTOS, ISABEL, R |
| description | Agente quelante de la fórmula general: **(Ver fórmula)** en la que m es 0 ó 1 X es NR4; Y es NHR5, SR5 o P(R5)2; R1 y R3 son iguales o diferentes y se seleccionan entre H, alquilo o arilo; R2 es H, COOH, NHR6 o (CH2)nCOOR6; R4 es (CH2)nCOOR6, o (CH2)nOR6; R5 es H, alquilo, arilo, (CH2) nCOOR6, o (CH2)nOR6; R6 es H, alquilo, arilo o una biomolécula; y n es 1,2, 3, 4, 5, 6, 7, 8, 9 ó 10.
The present invention relates to a chelating agent of the general formula: (I), wherein m is 0 or 1; X is NR4 or S; Y is SR5, NHR5 or P(R5)2; R1 and R3 are the same or different and are selected from H, alkyl or aryl; R2 is H, COOH, NHR6 or (CH2)nCOOR6; R4 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6; R5 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6, R6 is H, alkyl or aryl; n is 1, 2, 3, 4, 5, 6, 7, 8, 9 or 10; and when R1=R3=CH3, R2, R4 and R5 are not all three H. The invention further relates to a method and kit for the preparation of radiolabeled biomolecules while using the chelating agent. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_ES2346974TT3</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>ES2346974TT3</sourcerecordid><originalsourceid>FETCH-epo_espacenet_ES2346974TT33</originalsourceid><addsrcrecordid>eNqNjLEKwkAQRNNYiPoPa6-NFxTLy91GVy578bIptAlRzko0EP8fE_ADrIZ5zJtpcisp6Kt35DxIIIss2nrIKK_ZkGft4FwjGM9CyAiODpqtr6DUQQ-4KB2ehmpx1I0OmefxK-AKxMAFCp4nk0f77OPil7NkmaOY4zp27yb2XXuPr_hpsNqodLvfpSJK_bP5AvV9NE4</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>PIRAZOLILO TRIDENTADO BIFUNCIONAL QUE CONTIENE LIGANDOS PARA COMPLEJOS DE TRICARBONILO RE, TC Y MN</title><source>esp@cenet</source><creator>ROCHA PAULO, ANTONIO, M ; GALAMBA CORREIA, JOAO, D ; ALVES, SUSANA ; VITOR, RUTE ; SANTOS, ISABEL, R</creator><creatorcontrib>ROCHA PAULO, ANTONIO, M ; GALAMBA CORREIA, JOAO, D ; ALVES, SUSANA ; VITOR, RUTE ; SANTOS, ISABEL, R</creatorcontrib><description>Agente quelante de la fórmula general: **(Ver fórmula)** en la que m es 0 ó 1 X es NR4; Y es NHR5, SR5 o P(R5)2; R1 y R3 son iguales o diferentes y se seleccionan entre H, alquilo o arilo; R2 es H, COOH, NHR6 o (CH2)nCOOR6; R4 es (CH2)nCOOR6, o (CH2)nOR6; R5 es H, alquilo, arilo, (CH2) nCOOR6, o (CH2)nOR6; R6 es H, alquilo, arilo o una biomolécula; y n es 1,2, 3, 4, 5, 6, 7, 8, 9 ó 10.
The present invention relates to a chelating agent of the general formula: (I), wherein m is 0 or 1; X is NR4 or S; Y is SR5, NHR5 or P(R5)2; R1 and R3 are the same or different and are selected from H, alkyl or aryl; R2 is H, COOH, NHR6 or (CH2)nCOOR6; R4 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6; R5 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6, R6 is H, alkyl or aryl; n is 1, 2, 3, 4, 5, 6, 7, 8, 9 or 10; and when R1=R3=CH3, R2, R4 and R5 are not all three H. The invention further relates to a method and kit for the preparation of radiolabeled biomolecules while using the chelating agent.</description><language>spa</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2010</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20101022&DB=EPODOC&CC=ES&NR=2346974T3$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20101022&DB=EPODOC&CC=ES&NR=2346974T3$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>ROCHA PAULO, ANTONIO, M</creatorcontrib><creatorcontrib>GALAMBA CORREIA, JOAO, D</creatorcontrib><creatorcontrib>ALVES, SUSANA</creatorcontrib><creatorcontrib>VITOR, RUTE</creatorcontrib><creatorcontrib>SANTOS, ISABEL, R</creatorcontrib><title>PIRAZOLILO TRIDENTADO BIFUNCIONAL QUE CONTIENE LIGANDOS PARA COMPLEJOS DE TRICARBONILO RE, TC Y MN</title><description>Agente quelante de la fórmula general: **(Ver fórmula)** en la que m es 0 ó 1 X es NR4; Y es NHR5, SR5 o P(R5)2; R1 y R3 son iguales o diferentes y se seleccionan entre H, alquilo o arilo; R2 es H, COOH, NHR6 o (CH2)nCOOR6; R4 es (CH2)nCOOR6, o (CH2)nOR6; R5 es H, alquilo, arilo, (CH2) nCOOR6, o (CH2)nOR6; R6 es H, alquilo, arilo o una biomolécula; y n es 1,2, 3, 4, 5, 6, 7, 8, 9 ó 10.
The present invention relates to a chelating agent of the general formula: (I), wherein m is 0 or 1; X is NR4 or S; Y is SR5, NHR5 or P(R5)2; R1 and R3 are the same or different and are selected from H, alkyl or aryl; R2 is H, COOH, NHR6 or (CH2)nCOOR6; R4 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6; R5 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6, R6 is H, alkyl or aryl; n is 1, 2, 3, 4, 5, 6, 7, 8, 9 or 10; and when R1=R3=CH3, R2, R4 and R5 are not all three H. The invention further relates to a method and kit for the preparation of radiolabeled biomolecules while using the chelating agent.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2010</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNjLEKwkAQRNNYiPoPa6-NFxTLy91GVy578bIptAlRzko0EP8fE_ADrIZ5zJtpcisp6Kt35DxIIIss2nrIKK_ZkGft4FwjGM9CyAiODpqtr6DUQQ-4KB2ehmpx1I0OmefxK-AKxMAFCp4nk0f77OPil7NkmaOY4zp27yb2XXuPr_hpsNqodLvfpSJK_bP5AvV9NE4</recordid><startdate>20101022</startdate><enddate>20101022</enddate><creator>ROCHA PAULO, ANTONIO, M</creator><creator>GALAMBA CORREIA, JOAO, D</creator><creator>ALVES, SUSANA</creator><creator>VITOR, RUTE</creator><creator>SANTOS, ISABEL, R</creator><scope>EVB</scope></search><sort><creationdate>20101022</creationdate><title>PIRAZOLILO TRIDENTADO BIFUNCIONAL QUE CONTIENE LIGANDOS PARA COMPLEJOS DE TRICARBONILO RE, TC Y MN</title><author>ROCHA PAULO, ANTONIO, M ; GALAMBA CORREIA, JOAO, D ; ALVES, SUSANA ; VITOR, RUTE ; SANTOS, ISABEL, R</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_ES2346974TT33</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>spa</language><creationdate>2010</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>ROCHA PAULO, ANTONIO, M</creatorcontrib><creatorcontrib>GALAMBA CORREIA, JOAO, D</creatorcontrib><creatorcontrib>ALVES, SUSANA</creatorcontrib><creatorcontrib>VITOR, RUTE</creatorcontrib><creatorcontrib>SANTOS, ISABEL, R</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>ROCHA PAULO, ANTONIO, M</au><au>GALAMBA CORREIA, JOAO, D</au><au>ALVES, SUSANA</au><au>VITOR, RUTE</au><au>SANTOS, ISABEL, R</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>PIRAZOLILO TRIDENTADO BIFUNCIONAL QUE CONTIENE LIGANDOS PARA COMPLEJOS DE TRICARBONILO RE, TC Y MN</title><date>2010-10-22</date><risdate>2010</risdate><abstract>Agente quelante de la fórmula general: **(Ver fórmula)** en la que m es 0 ó 1 X es NR4; Y es NHR5, SR5 o P(R5)2; R1 y R3 son iguales o diferentes y se seleccionan entre H, alquilo o arilo; R2 es H, COOH, NHR6 o (CH2)nCOOR6; R4 es (CH2)nCOOR6, o (CH2)nOR6; R5 es H, alquilo, arilo, (CH2) nCOOR6, o (CH2)nOR6; R6 es H, alquilo, arilo o una biomolécula; y n es 1,2, 3, 4, 5, 6, 7, 8, 9 ó 10.
The present invention relates to a chelating agent of the general formula: (I), wherein m is 0 or 1; X is NR4 or S; Y is SR5, NHR5 or P(R5)2; R1 and R3 are the same or different and are selected from H, alkyl or aryl; R2 is H, COOH, NHR6 or (CH2)nCOOR6; R4 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6; R5 is H, alkyl, aryl, (CH2)nCOOR6 or (CH2)nOR6, R6 is H, alkyl or aryl; n is 1, 2, 3, 4, 5, 6, 7, 8, 9 or 10; and when R1=R3=CH3, R2, R4 and R5 are not all three H. The invention further relates to a method and kit for the preparation of radiolabeled biomolecules while using the chelating agent.</abstract><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | spa |
| recordid | cdi_epo_espacenet_ES2346974TT3 |
| source | esp@cenet |
| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | PIRAZOLILO TRIDENTADO BIFUNCIONAL QUE CONTIENE LIGANDOS PARA COMPLEJOS DE TRICARBONILO RE, TC Y MN |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-01-04T13%3A54%3A02IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=ROCHA%20PAULO,%20ANTONIO,%20M&rft.date=2010-10-22&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EES2346974TT3%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |