SOLID FORM OF A BRADYKININ B2-RECEPTOR ANTAGONIST

SOLID FORM OF A BRADYKININ B2-RECEPTOR ANTAGONIST

This invention relates to a solid form of the bradykinin (BK) B2-receptor antagonist (S)-N-(1-deutero-1-(3-chloro-5-fluoro-2-((2-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)quinolin-8-yloxy)methyl)phenyl)ethyl)-2-(difluoromethoxy)acetamide, pharmaceutical compositions comprising the solid form, and to...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
1. Verfasser: GIBSON, Christoph
Format: Patent
Sprache:eng ; fre ; ger
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
Beschreibung
Zusammenfassung:This invention relates to a solid form of the bradykinin (BK) B2-receptor antagonist (S)-N-(1-deutero-1-(3-chloro-5-fluoro-2-((2-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)quinolin-8-yloxy)methyl)phenyl)ethyl)-2-(difluoromethoxy)acetamide, pharmaceutical compositions comprising the solid form, and to methods of use thereof in the preparation of a pharmaceutical formulation and in treatment, prevention or management of diseases or conditions susceptible to treatment with a BK B2-receptor antagonist.