PRODUCTION METHOD FOR 2-FLUORO-4-BORONO-L-PHENYLALANINE, AND PRECURSOR OF 2-FLUORO-4-BORONO-L-PHENYLALANINE

The present invention involves preparing compounds represented by the formula. (In the formula: R 1 represents a Br group, an iodine group, a Cl group, an NO 2 group, or an NH 2 group; R 2 represents a halogen group, an NO 2 group, an NH 2 group, Sn(R 6 ) 3 , N=N-NR 7 R 8 , OSO 2 R 9 , N R 10 R 11 ,...

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Hauptverfasser: ISHINO, Yuko, UEHARA, Kohki, TAKENAKA, Hiroshi, TAGUCHI, Yusuke, YOSHIKAWA, Tomohiro, UEDA, Sayuri, NAKASHIMA, Hideki, KIRIHATA, Mitsunori, OHTA, Yoichiro
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creator ISHINO, Yuko
UEHARA, Kohki
TAKENAKA, Hiroshi
TAGUCHI, Yusuke
YOSHIKAWA, Tomohiro
UEDA, Sayuri
NAKASHIMA, Hideki
KIRIHATA, Mitsunori
OHTA, Yoichiro
description The present invention involves preparing compounds represented by the formula. (In the formula: R 1 represents a Br group, an iodine group, a Cl group, an NO 2 group, or an NH 2 group; R 2 represents a halogen group, an NO 2 group, an NH 2 group, Sn(R 6 ) 3 , N=N-NR 7 R 8 , OSO 2 R 9 , N R 10 R 11 , phenyliodonium, a heterocyclic group iodine, boric acid, or a borate ester; R 30 represents a protective group PG 1 ; R 40 or R 50 represent hydrogen, a protective group PG 2 , or C 6 H 5 (C 6 H 5 )C=N, wherein NR 40 R 50 are together.)
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subjects ACYCLIC OR CARBOCYCLIC COMPOUNDS
ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
APPARATUS THEREFOR
CHEMISTRY
GENERAL METHODS OF ORGANIC CHEMISTRY
METALLURGY
ORGANIC CHEMISTRY
title PRODUCTION METHOD FOR 2-FLUORO-4-BORONO-L-PHENYLALANINE, AND PRECURSOR OF 2-FLUORO-4-BORONO-L-PHENYLALANINE
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