PRODUCTION METHOD FOR 2-FLUORO-4-BORONO-L-PHENYLALANINE, AND PRECURSOR OF 2-FLUORO-4-BORONO-L-PHENYLALANINE

The present invention involves preparing compounds represented by the formula. (In the formula: R 1 represents a Br group, an iodine group, a Cl group, an NO 2 group, or an NH 2 group; R 2 represents a halogen group, an NO 2 group, an NH 2 group, Sn(R 6 ) 3 , N=N-NR 7 R 8 , OSO 2 R 9 , N R 10 R 11 ,...

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Bibliographische Detailangaben
Hauptverfasser: ISHINO, Yuko, UEHARA, Kohki, TAKENAKA, Hiroshi, TAGUCHI, Yusuke, YOSHIKAWA, Tomohiro, UEDA, Sayuri, NAKASHIMA, Hideki, KIRIHATA, Mitsunori, OHTA, Yoichiro
Format: Patent
Sprache:eng ; fre ; ger
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Zusammenfassung:The present invention involves preparing compounds represented by the formula. (In the formula: R 1 represents a Br group, an iodine group, a Cl group, an NO 2 group, or an NH 2 group; R 2 represents a halogen group, an NO 2 group, an NH 2 group, Sn(R 6 ) 3 , N=N-NR 7 R 8 , OSO 2 R 9 , N R 10 R 11 , phenyliodonium, a heterocyclic group iodine, boric acid, or a borate ester; R 30 represents a protective group PG 1 ; R 40 or R 50 represent hydrogen, a protective group PG 2 , or C 6 H 5 (C 6 H 5 )C=N, wherein NR 40 R 50 are together.)