A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST
The present invention is directed to a 2,6-substituted-4-monosubstitutedamino-pyrimidine compound of formula (I): or an enantiomer thereof, or an ester prodrug or a pharmaceutically acceptable salt thereof, or a pharmaceutical composition comprising such a compound. The invention also includes a met...
Gespeichert in:
Hauptverfasser: | , , , , , , , |
---|---|
Format: | Patent |
Sprache: | eng ; fre ; ger |
Schlagworte: | |
Online-Zugang: | Volltext bestellen |
Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
container_end_page | |
---|---|
container_issue | |
container_start_page | |
container_title | |
container_volume | |
creator | STOKLOSA, GREGORY T AGUIAR, JOACY C SHUM, PATRICK WAI-KWOK POLI, GREGORY B ZHAO, ZHICHENG HARRIS, KEITH JOHN CHOI-SLEDESKI, YONG-MI REILING, STEPHAN |
description | The present invention is directed to a 2,6-substituted-4-monosubstitutedamino-pyrimidine compound of formula (I): or an enantiomer thereof, or an ester prodrug or a pharmaceutically acceptable salt thereof, or a pharmaceutical composition comprising such a compound. The invention also includes a method of treatment of a patient by the administration of a pharmaceutically effective amount of such a compound. |
format | Patent |
fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_EP2547673A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>EP2547673A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_EP2547673A13</originalsourceid><addsrcrecordid>eNrjZHByVAgOdQoO8QwJDXF1UQiIDPL09XTx9HNVcAxWcFQICPIPDnF093H0A4opuBgpBLk6uwaE-AcpOPoBxf39PINDeBhY0xJzilN5oTQ3g4Kba4izh25qQX58anFBYnJqXmpJvGuAkamJuZm5saOhMRFKALZ3Ku0</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST</title><source>esp@cenet</source><creator>STOKLOSA, GREGORY T ; AGUIAR, JOACY C ; SHUM, PATRICK WAI-KWOK ; POLI, GREGORY B ; ZHAO, ZHICHENG ; HARRIS, KEITH JOHN ; CHOI-SLEDESKI, YONG-MI ; REILING, STEPHAN</creator><creatorcontrib>STOKLOSA, GREGORY T ; AGUIAR, JOACY C ; SHUM, PATRICK WAI-KWOK ; POLI, GREGORY B ; ZHAO, ZHICHENG ; HARRIS, KEITH JOHN ; CHOI-SLEDESKI, YONG-MI ; REILING, STEPHAN</creatorcontrib><description>The present invention is directed to a 2,6-substituted-4-monosubstitutedamino-pyrimidine compound of formula (I): or an enantiomer thereof, or an ester prodrug or a pharmaceutically acceptable salt thereof, or a pharmaceutical composition comprising such a compound. The invention also includes a method of treatment of a patient by the administration of a pharmaceutically effective amount of such a compound.</description><language>eng ; fre ; ger</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2013</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20130123&DB=EPODOC&CC=EP&NR=2547673A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20130123&DB=EPODOC&CC=EP&NR=2547673A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>STOKLOSA, GREGORY T</creatorcontrib><creatorcontrib>AGUIAR, JOACY C</creatorcontrib><creatorcontrib>SHUM, PATRICK WAI-KWOK</creatorcontrib><creatorcontrib>POLI, GREGORY B</creatorcontrib><creatorcontrib>ZHAO, ZHICHENG</creatorcontrib><creatorcontrib>HARRIS, KEITH JOHN</creatorcontrib><creatorcontrib>CHOI-SLEDESKI, YONG-MI</creatorcontrib><creatorcontrib>REILING, STEPHAN</creatorcontrib><title>A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST</title><description>The present invention is directed to a 2,6-substituted-4-monosubstitutedamino-pyrimidine compound of formula (I): or an enantiomer thereof, or an ester prodrug or a pharmaceutically acceptable salt thereof, or a pharmaceutical composition comprising such a compound. The invention also includes a method of treatment of a patient by the administration of a pharmaceutically effective amount of such a compound.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2013</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZHByVAgOdQoO8QwJDXF1UQiIDPL09XTx9HNVcAxWcFQICPIPDnF093H0A4opuBgpBLk6uwaE-AcpOPoBxf39PINDeBhY0xJzilN5oTQ3g4Kba4izh25qQX58anFBYnJqXmpJvGuAkamJuZm5saOhMRFKALZ3Ku0</recordid><startdate>20130123</startdate><enddate>20130123</enddate><creator>STOKLOSA, GREGORY T</creator><creator>AGUIAR, JOACY C</creator><creator>SHUM, PATRICK WAI-KWOK</creator><creator>POLI, GREGORY B</creator><creator>ZHAO, ZHICHENG</creator><creator>HARRIS, KEITH JOHN</creator><creator>CHOI-SLEDESKI, YONG-MI</creator><creator>REILING, STEPHAN</creator><scope>EVB</scope></search><sort><creationdate>20130123</creationdate><title>A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST</title><author>STOKLOSA, GREGORY T ; AGUIAR, JOACY C ; SHUM, PATRICK WAI-KWOK ; POLI, GREGORY B ; ZHAO, ZHICHENG ; HARRIS, KEITH JOHN ; CHOI-SLEDESKI, YONG-MI ; REILING, STEPHAN</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_EP2547673A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre ; ger</language><creationdate>2013</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>STOKLOSA, GREGORY T</creatorcontrib><creatorcontrib>AGUIAR, JOACY C</creatorcontrib><creatorcontrib>SHUM, PATRICK WAI-KWOK</creatorcontrib><creatorcontrib>POLI, GREGORY B</creatorcontrib><creatorcontrib>ZHAO, ZHICHENG</creatorcontrib><creatorcontrib>HARRIS, KEITH JOHN</creatorcontrib><creatorcontrib>CHOI-SLEDESKI, YONG-MI</creatorcontrib><creatorcontrib>REILING, STEPHAN</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>STOKLOSA, GREGORY T</au><au>AGUIAR, JOACY C</au><au>SHUM, PATRICK WAI-KWOK</au><au>POLI, GREGORY B</au><au>ZHAO, ZHICHENG</au><au>HARRIS, KEITH JOHN</au><au>CHOI-SLEDESKI, YONG-MI</au><au>REILING, STEPHAN</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST</title><date>2013-01-23</date><risdate>2013</risdate><abstract>The present invention is directed to a 2,6-substituted-4-monosubstitutedamino-pyrimidine compound of formula (I): or an enantiomer thereof, or an ester prodrug or a pharmaceutically acceptable salt thereof, or a pharmaceutical composition comprising such a compound. The invention also includes a method of treatment of a patient by the administration of a pharmaceutically effective amount of such a compound.</abstract><oa>free_for_read</oa></addata></record> |
fulltext | fulltext_linktorsrc |
identifier | |
ispartof | |
issn | |
language | eng ; fre ; ger |
recordid | cdi_epo_espacenet_EP2547673A1 |
source | esp@cenet |
subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
title | A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST |
url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-01-01T17%3A20%3A47IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=STOKLOSA,%20GREGORY%20T&rft.date=2013-01-23&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EEP2547673A1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |