Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors
Pyridine and pyrimidine compounds, and compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obse...
Gespeichert in:
| Hauptverfasser: | , , , , , , , , , , , , , , , , , , , |
|---|---|
| Format: | Patent |
| Sprache: | eng ; fre ; ger |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | RUMFELT, SHANNON SHAM, KELVIN CHEN, NING DEMORIN, FRENEL FILS ALLEN, JENNIFER R HARRINGTON, PAUL KALLER, MATTHEW R MONENSCHEIN, HOLGER RZASA, ROB BISWAS, KAUSTAV CHAVEZ, FRANK, JR HORNE, DAN YAO, GUOMIN FROHN, MIKE KUNZ, ROXANNE REICHELT, ANDREAS FALSEY, JAMES R PICKRELL, ALEX HU, ESSA NGUYEN, TOM |
| description | Pyridine and pyrimidine compounds, and compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_EP2364306B1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>EP2364306B1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_EP2364306B13</originalsourceid><addsrcrecordid>eNrjZHALqCzKTMnMS1VIzEtRKAByciHclNSizLLEksyy1GKFxGKFgoz8YiBOyUwtLkktSixOVTA0UMjMy8hMyizJLyrmYWBNS8wpTuWF0twMCm6uIc4euqkF-fGpxQWJyal5qSXxrgFGxmYmxgZmTobGRCgBAAOgM5g</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors</title><source>esp@cenet</source><creator>RUMFELT, SHANNON ; SHAM, KELVIN ; CHEN, NING ; DEMORIN, FRENEL FILS ; ALLEN, JENNIFER R ; HARRINGTON, PAUL ; KALLER, MATTHEW R ; MONENSCHEIN, HOLGER ; RZASA, ROB ; BISWAS, KAUSTAV ; CHAVEZ, FRANK, JR ; HORNE, DAN ; YAO, GUOMIN ; FROHN, MIKE ; KUNZ, ROXANNE ; REICHELT, ANDREAS ; FALSEY, JAMES R ; PICKRELL, ALEX ; HU, ESSA ; NGUYEN, TOM</creator><creatorcontrib>RUMFELT, SHANNON ; SHAM, KELVIN ; CHEN, NING ; DEMORIN, FRENEL FILS ; ALLEN, JENNIFER R ; HARRINGTON, PAUL ; KALLER, MATTHEW R ; MONENSCHEIN, HOLGER ; RZASA, ROB ; BISWAS, KAUSTAV ; CHAVEZ, FRANK, JR ; HORNE, DAN ; YAO, GUOMIN ; FROHN, MIKE ; KUNZ, ROXANNE ; REICHELT, ANDREAS ; FALSEY, JAMES R ; PICKRELL, ALEX ; HU, ESSA ; NGUYEN, TOM</creatorcontrib><description>Pyridine and pyrimidine compounds, and compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like.</description><language>eng ; fre ; ger</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2013</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20130424&DB=EPODOC&CC=EP&NR=2364306B1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20130424&DB=EPODOC&CC=EP&NR=2364306B1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>RUMFELT, SHANNON</creatorcontrib><creatorcontrib>SHAM, KELVIN</creatorcontrib><creatorcontrib>CHEN, NING</creatorcontrib><creatorcontrib>DEMORIN, FRENEL FILS</creatorcontrib><creatorcontrib>ALLEN, JENNIFER R</creatorcontrib><creatorcontrib>HARRINGTON, PAUL</creatorcontrib><creatorcontrib>KALLER, MATTHEW R</creatorcontrib><creatorcontrib>MONENSCHEIN, HOLGER</creatorcontrib><creatorcontrib>RZASA, ROB</creatorcontrib><creatorcontrib>BISWAS, KAUSTAV</creatorcontrib><creatorcontrib>CHAVEZ, FRANK, JR</creatorcontrib><creatorcontrib>HORNE, DAN</creatorcontrib><creatorcontrib>YAO, GUOMIN</creatorcontrib><creatorcontrib>FROHN, MIKE</creatorcontrib><creatorcontrib>KUNZ, ROXANNE</creatorcontrib><creatorcontrib>REICHELT, ANDREAS</creatorcontrib><creatorcontrib>FALSEY, JAMES R</creatorcontrib><creatorcontrib>PICKRELL, ALEX</creatorcontrib><creatorcontrib>HU, ESSA</creatorcontrib><creatorcontrib>NGUYEN, TOM</creatorcontrib><title>Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors</title><description>Pyridine and pyrimidine compounds, and compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2013</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZHALqCzKTMnMS1VIzEtRKAByciHclNSizLLEksyy1GKFxGKFgoz8YiBOyUwtLkktSixOVTA0UMjMy8hMyizJLyrmYWBNS8wpTuWF0twMCm6uIc4euqkF-fGpxQWJyal5qSXxrgFGxmYmxgZmTobGRCgBAAOgM5g</recordid><startdate>20130424</startdate><enddate>20130424</enddate><creator>RUMFELT, SHANNON</creator><creator>SHAM, KELVIN</creator><creator>CHEN, NING</creator><creator>DEMORIN, FRENEL FILS</creator><creator>ALLEN, JENNIFER R</creator><creator>HARRINGTON, PAUL</creator><creator>KALLER, MATTHEW R</creator><creator>MONENSCHEIN, HOLGER</creator><creator>RZASA, ROB</creator><creator>BISWAS, KAUSTAV</creator><creator>CHAVEZ, FRANK, JR</creator><creator>HORNE, DAN</creator><creator>YAO, GUOMIN</creator><creator>FROHN, MIKE</creator><creator>KUNZ, ROXANNE</creator><creator>REICHELT, ANDREAS</creator><creator>FALSEY, JAMES R</creator><creator>PICKRELL, ALEX</creator><creator>HU, ESSA</creator><creator>NGUYEN, TOM</creator><scope>EVB</scope></search><sort><creationdate>20130424</creationdate><title>Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors</title><author>RUMFELT, SHANNON ; SHAM, KELVIN ; CHEN, NING ; DEMORIN, FRENEL FILS ; ALLEN, JENNIFER R ; HARRINGTON, PAUL ; KALLER, MATTHEW R ; MONENSCHEIN, HOLGER ; RZASA, ROB ; BISWAS, KAUSTAV ; CHAVEZ, FRANK, JR ; HORNE, DAN ; YAO, GUOMIN ; FROHN, MIKE ; KUNZ, ROXANNE ; REICHELT, ANDREAS ; FALSEY, JAMES R ; PICKRELL, ALEX ; HU, ESSA ; NGUYEN, TOM</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_EP2364306B13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre ; ger</language><creationdate>2013</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>RUMFELT, SHANNON</creatorcontrib><creatorcontrib>SHAM, KELVIN</creatorcontrib><creatorcontrib>CHEN, NING</creatorcontrib><creatorcontrib>DEMORIN, FRENEL FILS</creatorcontrib><creatorcontrib>ALLEN, JENNIFER R</creatorcontrib><creatorcontrib>HARRINGTON, PAUL</creatorcontrib><creatorcontrib>KALLER, MATTHEW R</creatorcontrib><creatorcontrib>MONENSCHEIN, HOLGER</creatorcontrib><creatorcontrib>RZASA, ROB</creatorcontrib><creatorcontrib>BISWAS, KAUSTAV</creatorcontrib><creatorcontrib>CHAVEZ, FRANK, JR</creatorcontrib><creatorcontrib>HORNE, DAN</creatorcontrib><creatorcontrib>YAO, GUOMIN</creatorcontrib><creatorcontrib>FROHN, MIKE</creatorcontrib><creatorcontrib>KUNZ, ROXANNE</creatorcontrib><creatorcontrib>REICHELT, ANDREAS</creatorcontrib><creatorcontrib>FALSEY, JAMES R</creatorcontrib><creatorcontrib>PICKRELL, ALEX</creatorcontrib><creatorcontrib>HU, ESSA</creatorcontrib><creatorcontrib>NGUYEN, TOM</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>RUMFELT, SHANNON</au><au>SHAM, KELVIN</au><au>CHEN, NING</au><au>DEMORIN, FRENEL FILS</au><au>ALLEN, JENNIFER R</au><au>HARRINGTON, PAUL</au><au>KALLER, MATTHEW R</au><au>MONENSCHEIN, HOLGER</au><au>RZASA, ROB</au><au>BISWAS, KAUSTAV</au><au>CHAVEZ, FRANK, JR</au><au>HORNE, DAN</au><au>YAO, GUOMIN</au><au>FROHN, MIKE</au><au>KUNZ, ROXANNE</au><au>REICHELT, ANDREAS</au><au>FALSEY, JAMES R</au><au>PICKRELL, ALEX</au><au>HU, ESSA</au><au>NGUYEN, TOM</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors</title><date>2013-04-24</date><risdate>2013</risdate><abstract>Pyridine and pyrimidine compounds, and compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like.</abstract><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | eng ; fre ; ger |
| recordid | cdi_epo_espacenet_EP2364306B1 |
| source | esp@cenet |
| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-01-01T07%3A28%3A25IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=RUMFELT,%20SHANNON&rft.date=2013-04-24&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EEP2364306B1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |