AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS

This application relates to a compound of formula (I) (or a pharmaceutically acceptable salt of the compound or prodrug thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa and/or thrombin, as well as a process for its preparation and intermediate...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: ARGADE, ANKUSH, B, HERRON, DAVID, KENT, TEBBE, ANNE, LOUISE, WILEY, MICHAEL, ROBERT, GOODSON, THEODORE, JUNIOR, YEE, YING, KWONG, LEPORE, SALVATORE, DONATO, MENDEL, DAVID, MASTERS, JOHN, JOSEPH, SMITH, GERALD, FLOYD, MARQUART, ANGELA, LYNN, JOSEPH, SAJAN, RATZ, ANDREW, MICHAEL, MERRITT, LEANDER
Format: Patent
Sprache:eng ; fre ; ger
Schlagworte:
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
container_end_page
container_issue
container_start_page
container_title
container_volume
creator ARGADE, ANKUSH, B
HERRON, DAVID, KENT
TEBBE, ANNE, LOUISE
WILEY, MICHAEL, ROBERT
GOODSON, THEODORE, JUNIOR
YEE, YING, KWONG
LEPORE, SALVATORE, DONATO
MENDEL, DAVID
MASTERS, JOHN, JOSEPH
SMITH, GERALD, FLOYD
MARQUART, ANGELA, LYNN
JOSEPH, SAJAN
RATZ, ANDREW, MICHAEL
MERRITT, LEANDER
description This application relates to a compound of formula (I) (or a pharmaceutically acceptable salt of the compound or prodrug thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa and/or thrombin, as well as a process for its preparation and intermediates therefor. An example of a compound of formula (I) is (a).
format Patent
fullrecord <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_EP1817287B1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>EP1817287B1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_EP1817287B13</originalsourceid><addsrcrecordid>eNrjZLBwDPL3dQzxdFZwDfFwDVJwcQ3yDAPyw1yDFUKDXd1CfRQcgxVCPICqnDz9FDz9PDydPEP8g4J5GFjTEnOKU3mhNDeDgptriLOHbmpBfnxqcUFicmpeakm8a4ChhaG5kYW5k6ExEUoAMMQoYQ</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS</title><source>esp@cenet</source><creator>ARGADE, ANKUSH, B ; HERRON, DAVID, KENT ; TEBBE, ANNE, LOUISE ; WILEY, MICHAEL, ROBERT ; GOODSON, THEODORE, JUNIOR ; YEE, YING, KWONG ; LEPORE, SALVATORE, DONATO ; MENDEL, DAVID ; MASTERS, JOHN, JOSEPH ; SMITH, GERALD, FLOYD ; MARQUART, ANGELA, LYNN ; JOSEPH, SAJAN ; RATZ, ANDREW, MICHAEL ; MERRITT, LEANDER</creator><creatorcontrib>ARGADE, ANKUSH, B ; HERRON, DAVID, KENT ; TEBBE, ANNE, LOUISE ; WILEY, MICHAEL, ROBERT ; GOODSON, THEODORE, JUNIOR ; YEE, YING, KWONG ; LEPORE, SALVATORE, DONATO ; MENDEL, DAVID ; MASTERS, JOHN, JOSEPH ; SMITH, GERALD, FLOYD ; MARQUART, ANGELA, LYNN ; JOSEPH, SAJAN ; RATZ, ANDREW, MICHAEL ; MERRITT, LEANDER</creatorcontrib><description>This application relates to a compound of formula (I) (or a pharmaceutically acceptable salt of the compound or prodrug thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa and/or thrombin, as well as a process for its preparation and intermediates therefor. An example of a compound of formula (I) is (a).</description><language>eng ; fre ; ger</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2010</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20100210&amp;DB=EPODOC&amp;CC=EP&amp;NR=1817287B1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20100210&amp;DB=EPODOC&amp;CC=EP&amp;NR=1817287B1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>ARGADE, ANKUSH, B</creatorcontrib><creatorcontrib>HERRON, DAVID, KENT</creatorcontrib><creatorcontrib>TEBBE, ANNE, LOUISE</creatorcontrib><creatorcontrib>WILEY, MICHAEL, ROBERT</creatorcontrib><creatorcontrib>GOODSON, THEODORE, JUNIOR</creatorcontrib><creatorcontrib>YEE, YING, KWONG</creatorcontrib><creatorcontrib>LEPORE, SALVATORE, DONATO</creatorcontrib><creatorcontrib>MENDEL, DAVID</creatorcontrib><creatorcontrib>MASTERS, JOHN, JOSEPH</creatorcontrib><creatorcontrib>SMITH, GERALD, FLOYD</creatorcontrib><creatorcontrib>MARQUART, ANGELA, LYNN</creatorcontrib><creatorcontrib>JOSEPH, SAJAN</creatorcontrib><creatorcontrib>RATZ, ANDREW, MICHAEL</creatorcontrib><creatorcontrib>MERRITT, LEANDER</creatorcontrib><title>AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS</title><description>This application relates to a compound of formula (I) (or a pharmaceutically acceptable salt of the compound or prodrug thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa and/or thrombin, as well as a process for its preparation and intermediates therefor. An example of a compound of formula (I) is (a).</description><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2010</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZLBwDPL3dQzxdFZwDfFwDVJwcQ3yDAPyw1yDFUKDXd1CfRQcgxVCPICqnDz9FDz9PDydPEP8g4J5GFjTEnOKU3mhNDeDgptriLOHbmpBfnxqcUFicmpeakm8a4ChhaG5kYW5k6ExEUoAMMQoYQ</recordid><startdate>20100210</startdate><enddate>20100210</enddate><creator>ARGADE, ANKUSH, B</creator><creator>HERRON, DAVID, KENT</creator><creator>TEBBE, ANNE, LOUISE</creator><creator>WILEY, MICHAEL, ROBERT</creator><creator>GOODSON, THEODORE, JUNIOR</creator><creator>YEE, YING, KWONG</creator><creator>LEPORE, SALVATORE, DONATO</creator><creator>MENDEL, DAVID</creator><creator>MASTERS, JOHN, JOSEPH</creator><creator>SMITH, GERALD, FLOYD</creator><creator>MARQUART, ANGELA, LYNN</creator><creator>JOSEPH, SAJAN</creator><creator>RATZ, ANDREW, MICHAEL</creator><creator>MERRITT, LEANDER</creator><scope>EVB</scope></search><sort><creationdate>20100210</creationdate><title>AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS</title><author>ARGADE, ANKUSH, B ; HERRON, DAVID, KENT ; TEBBE, ANNE, LOUISE ; WILEY, MICHAEL, ROBERT ; GOODSON, THEODORE, JUNIOR ; YEE, YING, KWONG ; LEPORE, SALVATORE, DONATO ; MENDEL, DAVID ; MASTERS, JOHN, JOSEPH ; SMITH, GERALD, FLOYD ; MARQUART, ANGELA, LYNN ; JOSEPH, SAJAN ; RATZ, ANDREW, MICHAEL ; MERRITT, LEANDER</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_EP1817287B13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre ; ger</language><creationdate>2010</creationdate><topic>ACYCLIC OR CARBOCYCLIC COMPOUNDS</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>ARGADE, ANKUSH, B</creatorcontrib><creatorcontrib>HERRON, DAVID, KENT</creatorcontrib><creatorcontrib>TEBBE, ANNE, LOUISE</creatorcontrib><creatorcontrib>WILEY, MICHAEL, ROBERT</creatorcontrib><creatorcontrib>GOODSON, THEODORE, JUNIOR</creatorcontrib><creatorcontrib>YEE, YING, KWONG</creatorcontrib><creatorcontrib>LEPORE, SALVATORE, DONATO</creatorcontrib><creatorcontrib>MENDEL, DAVID</creatorcontrib><creatorcontrib>MASTERS, JOHN, JOSEPH</creatorcontrib><creatorcontrib>SMITH, GERALD, FLOYD</creatorcontrib><creatorcontrib>MARQUART, ANGELA, LYNN</creatorcontrib><creatorcontrib>JOSEPH, SAJAN</creatorcontrib><creatorcontrib>RATZ, ANDREW, MICHAEL</creatorcontrib><creatorcontrib>MERRITT, LEANDER</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>ARGADE, ANKUSH, B</au><au>HERRON, DAVID, KENT</au><au>TEBBE, ANNE, LOUISE</au><au>WILEY, MICHAEL, ROBERT</au><au>GOODSON, THEODORE, JUNIOR</au><au>YEE, YING, KWONG</au><au>LEPORE, SALVATORE, DONATO</au><au>MENDEL, DAVID</au><au>MASTERS, JOHN, JOSEPH</au><au>SMITH, GERALD, FLOYD</au><au>MARQUART, ANGELA, LYNN</au><au>JOSEPH, SAJAN</au><au>RATZ, ANDREW, MICHAEL</au><au>MERRITT, LEANDER</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS</title><date>2010-02-10</date><risdate>2010</risdate><abstract>This application relates to a compound of formula (I) (or a pharmaceutically acceptable salt of the compound or prodrug thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa and/or thrombin, as well as a process for its preparation and intermediates therefor. An example of a compound of formula (I) is (a).</abstract><oa>free_for_read</oa></addata></record>
fulltext fulltext_linktorsrc
identifier
ispartof
issn
language eng ; fre ; ger
recordid cdi_epo_espacenet_EP1817287B1
source esp@cenet
subjects ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title AROMATIC ETHER DERIVATIVES USEFUL AS THROMBIN INHIBITORS
url https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2024-12-25T06%3A32%3A53IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=ARGADE,%20ANKUSH,%20B&rft.date=2010-02-10&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EEP1817287B1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true