PROCESSES FOR THE PREPARATION OF (R)-G(A)-(2,3-DIMETHOXYPHENYL)-1-(2-(4-FLUOROPHENYL)ETHYL)-4-PIPERIDINEMETHANOL
The present invention provides various processes for the preparation of (R)-±-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol. These processes may be characterized by the following scheme:
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| creator | HAWTORNE ROBERT A MINISH, SHARON K SKULTETY PAUL F DAUGS, EDWARD D BINA ALAN G ORTYL THOMAS T HITT JAMES E FLEMMING HANS-WOLFRAM RAJEWSKI LIAN G SACK MARVIN J HILPERT THOMAS H.E STOLTZ-DUNN SANDRA K EVANS JONATHAN C GUILLAMOT GERARD KING CHI-HSIN R TIGNER ALONZO L KOEK JOHANNES N MARGOLIN ALEXEY L LASKOVICS FREDERICK M LEFLER JOHN M |
| description | The present invention provides various processes for the preparation of (R)-±-(2,3-dimethoxyphenyl)-1-[2-(4-fluorophenyl)ethyl]-4-piperidinemethanol. These processes may be characterized by the following scheme: |
| format | Patent |
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These processes may be characterized by the following scheme:</abstract><edition>7</edition><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | PROCESSES FOR THE PREPARATION OF (R)-G(A)-(2,3-DIMETHOXYPHENYL)-1-(2-(4-FLUOROPHENYL)ETHYL)-4-PIPERIDINEMETHANOL |
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