Process for preparing epibatidine

The subject-matter of the invention is a process for preparing racemic or optically active epibatidine of formula which comprises cyclising a 1-ÄdiacylaminoÜ-2-Ä6'-chloro)-pyrid-3'-ylÜ-4-ÄaminoÜ-cyclohexane of general formula wherein Ac stands for an acyl group. The advantage of the proces...

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Bibliographische Detailangaben
Hauptverfasser:	GIGLER, GABOR, SIMIG, GYULA, DRABANT, SANDOR, TEMESVARI NEE MAJOR, ESZTER, BLASK , GABOR, FEKETE, MARTON, BALOGH NEE KARDOS, ZSUZSANNA, MANDI, ATTILA, SZANTAY, CSABA, LAX, GYOERGYI, SZALLASI, TAMAS, SZANTAY JR., CSABA, MOLDVAI, ISTVAN
Format:	Patent
Sprache:	eng ; fre ; ger
Schlagworte:	CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:	The subject-matter of the invention is a process for preparing racemic or optically active epibatidine of formula which comprises cyclising a 1-ÄdiacylaminoÜ-2-Ä6'-chloro)-pyrid-3'-ylÜ-4-ÄaminoÜ-cyclohexane of general formula wherein Ac stands for an acyl group. The advantage of the process is that readily available starting materials are used and the procedure is suitable for industrial scale productions, too.