Stereoselective process for producing dihydro-2,3-benzodiazepine derivatives

A process for stereoselectively forming N-substituted dihydro-2,3 benzodiazepines of formula (I) which are useful as AMPA receptor antagonists, and novel intermediates useful in the process.

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: HANSEN, MARVIN MARTIN, VICENZI, JEFFREY THOMAS, VARIE, DAVID LEE, ANDERSON, BENJAMIN, ZMIJEWSKI, MILTON JOSEPH
Format: Patent
Sprache:eng ; fre ; ger
Schlagworte:
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
Beschreibung
Zusammenfassung:A process for stereoselectively forming N-substituted dihydro-2,3 benzodiazepines of formula (I) which are useful as AMPA receptor antagonists, and novel intermediates useful in the process.