VERFAHREN FÜR DIE HERSTELLUNG VON 4(5)-AMINO-5(4)-CARBOXAMIDOIMIDAZOLEN UND DEREN ZWISCHENPRODUKTE

The invention provides novel processes for preparing efficiently compounds of general formula (I) (wherein R1 and R2 are each independently hydrogen, optionally substituted C1-C10 alkyl, C3-C14 hydrocarbyl bearing an alicyclic skeleton, or the like) and intermediates thereof. Compounds of general fo...

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Hauptverfasser: SHIBASAKI, HIROAKI, TAKASE, MITSURU, ISHII, YUTAKA, NAGASAKI, FUMIHIKO, OOHATA, KIMIHIKO, YAMAZAKI, SATORU
Format: Patent
Sprache:ger
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Zusammenfassung:The invention provides novel processes for preparing efficiently compounds of general formula (I) (wherein R1 and R2 are each independently hydrogen, optionally substituted C1-C10 alkyl, C3-C14 hydrocarbyl bearing an alicyclic skeleton, or the like) and intermediates thereof. Compounds of general formula (I) can be prepared by subjecting compounds of general formula (II) and/or salts thereof to cyclization hydrolysis in an aqueous basic solution. Further, compounds of general formula (II) can be prepared from industrially easily available diaminomaleonitrile in a high yield.