2-imino-1,2-dihydro-3h-1,4-benzodiazepines

2-Imino-1,2-dihydro-3H-1,4-benzodiazepines. Title cpds. of formula (I): R1 = H, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or aralkyl (up to 12C); R2 = H, alkyl or benzyl, R3 = aryl, heteroaryl, alkyl, alkenyl, cycloalkyl or cycloalkenyl and opt. mono-substd. in the benzene ring of the ring s...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: HANSWILLI VON BRACHEL,DR, OTTO GRAEWINGER,DR, KLAUS RESAG,DR, ECKHARD SCHRAVEN,DR, ROLF-EBERHARD NITZ,DR.MED
Format: Patent
Sprache:eng ; ger
Schlagworte:
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
Beschreibung
Zusammenfassung:2-Imino-1,2-dihydro-3H-1,4-benzodiazepines. Title cpds. of formula (I): R1 = H, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or aralkyl (up to 12C); R2 = H, alkyl or benzyl, R3 = aryl, heteroaryl, alkyl, alkenyl, cycloalkyl or cycloalkenyl and opt. mono-substd. in the benzene ring of the ring system by halogen, alkyl, CF3, MeSO2, MeS, MeO or NO2 and disubstd. by halogen or alkyl are prepd. by cyclising O-R1NH.C6H4C(R3)=N.CH(R2).CN. (I) are sedatives, muscle relaxants, anxiolytic agents and anticonvulsants; certain (I) are novel.