2-imino-1,2-dihydro-3h-1,4-benzodiazepines
2-Imino-1,2-dihydro-3H-1,4-benzodiazepines. Title cpds. of formula (I): R1 = H, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or aralkyl (up to 12C); R2 = H, alkyl or benzyl, R3 = aryl, heteroaryl, alkyl, alkenyl, cycloalkyl or cycloalkenyl and opt. mono-substd. in the benzene ring of the ring s...
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Format: | Patent |
Sprache: | eng ; ger |
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Zusammenfassung: | 2-Imino-1,2-dihydro-3H-1,4-benzodiazepines. Title cpds. of formula (I): R1 = H, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl or aralkyl (up to 12C); R2 = H, alkyl or benzyl, R3 = aryl, heteroaryl, alkyl, alkenyl, cycloalkyl or cycloalkenyl and opt. mono-substd. in the benzene ring of the ring system by halogen, alkyl, CF3, MeSO2, MeS, MeO or NO2 and disubstd. by halogen or alkyl are prepd. by cyclising O-R1NH.C6H4C(R3)=N.CH(R2).CN. (I) are sedatives, muscle relaxants, anxiolytic agents and anticonvulsants; certain (I) are novel. |
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