5-VINYL-QUINOLONE-CARBOXYLIC, 5-VINYL-NAPHTHYRIDON-CARBOXYLIC, +5-ETHINYL-QUINOLONE-CARBOXYLIC AND 5-ETHINYL-NAPHTHYRIDON-CARBOXYLIC ACIDS, PROCESS OF THEIR PREPARATION, MEDICAMENTS IN WHICH SAID COMPOUNDS ARE COMPRISED AND THEIR USE

Quinolone and naphthyridone derivs. of formula (I), and their hydrates, acid addn. salts, and alkali-, alkaline earth, silver and guanidinium salts, are new. R1 = 1-4C alkyl (opt. substd. by OH, halo or 1-3C alkoxy), 3-6C cycloalkyl (opt. substd. by halo or 1-3C alkyl), 2-4C alkenyl, 1-3C alkoxy, am...

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Bibliographische Detailangaben
Hauptverfasser:	PETERSEN UWE DR, HIMMLER THOMAS DR, ENDERMANN RAINER DR, WETZSTEIN HEINZ-GEORG DR, BREMM KLAUS DIETER DR, STEGEMANN MICHAEL DR
Format:	Patent
Sprache:	eng
Schlagworte:	AGRICULTURE ANIMAL HUSBANDRY BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES CHEMISTRY FISHING FODDER FOODS OR FOODSTUFFS FOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BYSUBCLASSES A23B - A23J FORESTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HUNTING HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PEST REPELLANTS OR ATTRACTANTS PLANT GROWTH REGULATORS PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTSTHEREOF PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OFNUTRITIVE QUALITIES, PHYSICAL TREATMENT THEIR TREATMENT, NOT COVERED BY OTHER CLASSES TRAPPING
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Beschreibung
Zusammenfassung:	Quinolone and naphthyridone derivs. of formula (I), and their hydrates, acid addn. salts, and alkali-, alkaline earth, silver and guanidinium salts, are new. R1 = 1-4C alkyl (opt. substd. by OH, halo or 1-3C alkoxy), 3-6C cycloalkyl (opt. substd. by halo or 1-3C alkyl), 2-4C alkenyl, 1-3C alkoxy, amino, 1-3C monoalkylamino, 2-6C dialkylamino, or phenyl (opt. substd. by 1-3 halo); R2 = H, 1-4C alkyl or (5-methyl-2-oxo-1,3-dioxol-4-yl)-methyl; X = CH, C-halo, COMe, COCHF2, CMe or N; Z = CR4=CHR3 or C IDENTICAL CR5; R3 = H, 1-3C alkyl, 1-3C alkoxy, or 1-3C alkoxy-methyl; R4 = H or halo; R5 = H, 1-6C alkyl (opt. substd. by 1-3 halo or OH), 2-3C alkenyl, 1-3C alkoxy, 1-3C alkoxy-methyl, halo or SiMe3; R6 = H, 1-4C alkyl (opt. substd. by OH or OMe), cyclopropyl, 1-4C oxoalkyl, or 1-3C acyl; Y = NR'R"; NR'R" = pyrrolyl, imidazolyl or a specified satd. or mono-unsatd. mono-or bicyclic ring, (opt. contg. O or a second N, opt. substd.)