Process for preparing 4"-substituted derivatives of 9-deoxo-9a-aza-9a- homoerythromycin

The invention relates to processes for preparing compounds of formula 1 wherein R is as defined herein, and to pharmaceutically acceptable salts thereof, as well as intermediates useful in such processes. The compounds of formula 1 are antibacterial agents that may be used to treat various bacterial...

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Bibliographische Detailangaben
Hauptverfasser:	SKLAVOUNOS CONSTANTINE, LEHNER RICHARD SHELTON, TUCKER JOHN LLOYD, WEI LULIN, HAMMEN PHILIP DIETRICH, NEGRI JOANNA TERESA, MAHON KERRY PETER JR
Format:	Patent
Sprache:	cze ; eng
Schlagworte:	APPARATUS THEREFOR CHEMISTRY DERIVATIVES THEREOF GENERAL METHODS OF ORGANIC CHEMISTRY HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY NUCLEIC ACIDS NUCLEOSIDES NUCLEOTIDES ORGANIC CHEMISTRY SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS SUGARS
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Beschreibung
Zusammenfassung:	The invention relates to processes for preparing compounds of formula 1 wherein R is as defined herein, and to pharmaceutically acceptable salts thereof, as well as intermediates useful in such processes. The compounds of formula 1 are antibacterial agents that may be used to treat various bacterial and protozoa infections. The invention also relates to pharmaceutical compositions containing compounds prepared by the processes of the invention and to methods of treating bacterial protozoa infections by administering such compounds.