Novel crystals of 5-hydroxycarbamimidoyl-2-hydroxybenzenesulfonamide derivative

The present invention provides a novel crystalline form of n-butyl Ä4-Ä2-Ä2-hydroxy-5-(N-hydroxycarbamimidoyl) benzenesulfonylaminoÜethylÜ-2'-methanesulfonyl-3-yloxyÜ acetate hydrochloride, pharmaceutical compositions containing the same and their uses, which exhibits excellent inhibitory activ...

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Bibliographische Detailangaben
1. Verfasser:	MUKAIYAMA HARUNOBU,KAI YUICHIRO,TAKEUCHI HIDEKI,YOKOYAMA KENJI,TERAO YOSHIHIRO,AKAHANE SATOSHI
Format:	Patent
Sprache:	eng
Schlagworte:	ACYCLIC OR CARBOCYCLIC COMPOUNDS CHEMISTRY HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:	The present invention provides a novel crystalline form of n-butyl Ä4-Ä2-Ä2-hydroxy-5-(N-hydroxycarbamimidoyl) benzenesulfonylaminoÜethylÜ-2'-methanesulfonyl-3-yloxyÜ acetate hydrochloride, pharmaceutical compositions containing the same and their uses, which exhibits excellent inhibitory activities against activated blood coagulation factor X, and is useful for the treatment or prevention of a tromboembolic disease.