PI3K-alpha inhibitors and methods of use thereof

The present disclosure relates to novel compounds and pharmaceutical compositions thereof, and methods of inhibiting P13K-alpha enzyme activity using the compounds and compositions of the present disclosure. The present disclosure further relates to, but is not limited to, methods of treating condit...

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Hauptverfasser: UTHAN JESPER, MOHAMED TAMER, WALTERS WILLIAM P, BEARNEY AARON J, TANWELL KEVIN, KRUEGER ERIC B, VEMULA NARASIMHA, LESCARBO ANDREA, WANG QIGUI, TAYLOR ALEXANDER M, GIORDANETTO FRANCESCO, GALOZIA STEFANO, ATIENSA BAKHTIAR-JAN, KURUKULA SURIYA RAMESH, GIGUERE JEAN-BENOIT, PAHL MICHAEL, CHEN FEI, JOBIN-DESLAURIER AURELIEN, LANDAGARE ELENA, REINER KEVIN D, GUNAYDIN HAKAN, LEPUTTE THOMAS, SAURAT REGIS, BERTRAND-LAPIERLE MICKAEL, BOZIO ALBERTO, MCLEAN THOMAS H, DIPIETRO LUCIAN V, PAN YUE, LARIVE ALAIN, SCHOTTSREEVES KEITH C, MAERTENS GERRIT, PIERCE LINDA C. T, STURINO CHRISTOPHER, PESCHELSKY YVONNE, CITALE SALVATORE, FRIEDRICH CHRISTIAN G, DENINO MICHAEL P, ZHANG HANMO, BOUSQUET YVES, LI JUNYI, TANG YONG, MAEDER MORGAN M
Format: Patent
Sprache:chi ; eng
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