Tricyclic vasopressin agonists

本发明提供了通式(I)化合物:其中W是O或NH,可以被任意取代,以及利用这些化合物通过其后叶加压素激动剂活性,治疗或减轻有关疾病的方法和其药物组合物,其中所述病症包括尿崩症、夜间遗尿、夜尿症、尿失禁、出血和血凝固紊乱或不能暂时延迟排尿。∴ The present invention provides compounds of general formula (I): wherein W is O or NH, optionally substituted, as well as methods and pharmaceutical compositions utilising these co...

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Bibliographische Detailangaben
1. Verfasser: A. A. FAILLI,J. S. SHUMSKY,R. J. STEFFAN
Format: Patent
Sprache:chi ; eng
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Zusammenfassung:本发明提供了通式(I)化合物:其中W是O或NH,可以被任意取代,以及利用这些化合物通过其后叶加压素激动剂活性,治疗或减轻有关疾病的方法和其药物组合物,其中所述病症包括尿崩症、夜间遗尿、夜尿症、尿失禁、出血和血凝固紊乱或不能暂时延迟排尿。∴ The present invention provides compounds of general formula (I): wherein W is O or NH, optionally substituted, as well as methods and pharmaceutical compositions utilising these compounds for the treatment of disorder which may be remedied or alleviated by vasopressin agonist activity, including diabetes insipidus, nocturnal enuresis, nocturia, urinary incontinence, bleeding and coagulation disorders, or temporary delay of urination.