N-cyclohexyl-furan-2-formamide compound as well as preparation method and application thereof

N-cyclohexyl-furan-2-formamide compound as well as preparation method and application thereof

The invention discloses an N-cyclohexyl-furan-2-formamide compound as well as a preparation method and application of the N-cyclohexyl-furan-2-formamide compound. The N-cyclohexyl-furan-2-formamide compound can be used for preparing an anti-schizophrenia drug SIPI6398, and has the following remarkab...

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Hauptverfasser: CHEN XIAOWEN, LI JIANQI, SU XIAOJING, PU QIANG, QI YANGLI, ZHOU AINAN
Format: Patent
Sprache:chi ; eng
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CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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creator CHEN XIAOWEN
LI JIANQI
SU XIAOJING
PU QIANG
QI YANGLI
ZHOU AINAN
description The invention discloses an N-cyclohexyl-furan-2-formamide compound as well as a preparation method and application of the N-cyclohexyl-furan-2-formamide compound. The N-cyclohexyl-furan-2-formamide compound can be used for preparing an anti-schizophrenia drug SIPI6398, and has the following remarkable advantages compared with the prior art and reported literatures: 1, when the N-cyclohexyl-furan-2-formamide compound disclosed by the invention is used for synthesizing the SIPI6398 without the need of a reaction process of connecting a protecting group and removing the protecting group so that atom economy is high; 2, when the N-cyclohexyl-furan-2-formamide compound is used for preparing SIPI6398, the raw materials are cheap and easy to obtain, the cost is low, the reaction conditions are mild, the yield is stable, the operation is simple and convenient, the three-waste pollution is little, and the industrial production is easy, and the N-cyclohexyl-furan-2-formamide compound is a compound with the following st
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title N-cyclohexyl-furan-2-formamide compound as well as preparation method and application thereof
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