Synthesis method for 1-boralkylmethyl-6-aryl-3-benzenesulfonyl-3-azabicyclohexane derivative

The invention provides a synthesis method for a 1-boralkylmethyl-6-aryl-3-benzenesulfonyl-3-azabicyclohexane derivative. According to the invention, a target product is synthesized by taking an N-propargyl-N-(3-arylallyl)benzenesulfonamide derivative as a raw material, divalent palladium as a catalyst and bisdiboron as a boron reagent; and the structure of the target product is characterized and analyzed through methods of IR, 1H NMR, 13C NMR, HRMS and the like. The method provided by the invention has the advantages of easily available raw materials, simple operation, convenient subsequent treatment and the like. 本发明提供了一种1-硼烷基甲基-6-芳基-3-苯磺酰基-3-氮杂双环己烷衍生物的合成方法，以N-炔丙基-N-(3-芳基烯丙基)苯磺酰胺衍生物为原料，以二价钯为催化剂，联硼酸频那醇酯为硼试剂，合成得到目标产物，并对目标产物的结构通过IR、H NMR、C NMR和HRMS等方法进行了表征和分析。该方法具有原料易得、操作简单、后续处理方便等优点。