NEW PICOLINIC ACID DERIVATIVES AND THEIR USE AS INTERMEDIATES

NEW PICOLINIC ACID DERIVATIVES AND THEIR USE AS INTERMEDIATES

The present invention relates to new picolinic acid derivatives of formula (I) and their use as intermediates in the process of making pyridine derivatives, including (S)-3-amino-6- methoxy-N-(3,3,3-trifluoro-2-hydroxy-2-methylpropyl)-5-(trifluoromethyl)picolinamide that are useful for the treatment...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: HEINZ THOMAS, ZAUGG WERNER, MARTIN BENJAMIN, RAMPF FLORIAN ANDREAS
Format: Patent
Sprache:chi ; eng
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Beschreibung
Zusammenfassung:The present invention relates to new picolinic acid derivatives of formula (I) and their use as intermediates in the process of making pyridine derivatives, including (S)-3-amino-6- methoxy-N-(3,3,3-trifluoro-2-hydroxy-2-methylpropyl)-5-(trifluoromethyl)picolinamide that are useful for the treatment of respiratory disorders. (I) 本发明涉及具有式(I)的新的吡啶甲酸衍生物及其在制备可用于治疗呼吸障碍的吡啶衍生物的方法中作为中间体的用途，这些吡啶衍生物包括(S)-3-氨基-6-甲氧基-N-(3,3,3-三氟-2-羟基-2-甲基丙基)-5-(三氟甲基)吡啶甲酰胺。