Compuestos derivados de 1h-benzo[d]imidazol o sus sales; composicion farmaceutica; y uso en infecciones bacterianas

Compuestos derivados de 1h-benzo[d]imidazol o sus sales; composicion farmaceutica; y uso en infecciones bacterianas

The present invention relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof wherein X and R are as defined herein. The compounds of formula (I) are useful as gyrase and/or topoisomerase IV inhibitors for treating bacterial infections. The compounds of formula (I) either...

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Bibliographische Detailangaben
Hauptverfasser: GRILLOT ANNE-LAURE, BENNANI YOUSSEF LAAFIRET, O"DOWD HARDWIN, PEROLA EMANUELE, LE TIRAN ARNAUD, CHARIFSON PAUL
Format: Patent
Sprache:spa
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:The present invention relates to a compound of formula (I) or a pharmaceutically acceptable salt thereof wherein X and R are as defined herein. The compounds of formula (I) are useful as gyrase and/or topoisomerase IV inhibitors for treating bacterial infections. The compounds of formula (I) either possess a broad range of anti-bacterial activity and advantageous toxicological properties or are prodrugs of compounds having said activity.