SMALL MOLECULE INHIBITORS OF PBRM1-BD2
The present disclosure provides novel inhibitors of PBRM1, specifically the 2nd bromodomain of PBRM1 (PBRM1-BD2), pharmaceutical compositions and methods of use thereof. La présente invention concerne de nouveaux inhibiteurs de PBRM1, plus spécifiquement le 2ème bromodomaine de PBRM1 (PBRM1-BD2), de...
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| creator | SHISHODIA, SHIFALI SMITH, BRIAN CHRISTOPHER GOETZ, CHRISTOPHER J OLP, MICHAEL D |
| description | The present disclosure provides novel inhibitors of PBRM1, specifically the 2nd bromodomain of PBRM1 (PBRM1-BD2), pharmaceutical compositions and methods of use thereof.
La présente invention concerne de nouveaux inhibiteurs de PBRM1, plus spécifiquement le 2ème bromodomaine de PBRM1 (PBRM1-BD2), des compositions pharmaceutiques et leurs méthodes d'utilisation. |
| format | Patent |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | SMALL MOLECULE INHIBITORS OF PBRM1-BD2 |
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