IMIDAZO [4, 5 -C] QUINOLIN- 2 -ONE COMPOUND AND ITS USE AS PI3 KINASE / MTOR DUAL INHIBITOR

IMIDAZO [4, 5 -C] QUINOLIN- 2 -ONE COMPOUND AND ITS USE AS PI3 KINASE / MTOR DUAL INHIBITOR

The present invention provides an imidazo[4,5-c]quinolin-2-one compound (formula (I)), or a pharmaceutically acceptable salt thereof, that inhibits both PI3K and mTOR and, therefore, is useful in the treatment of cancer. La présente invention concerne un composé d'imidazo[4,5-c]quinolin-2-one (...

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Bibliographische Detailangaben
Hauptverfasser: MADER, MARY MARGARET, BARDA, DAVID ANTHONY
Format: Patent
Sprache:eng ; fre
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Zusammenfassung:The present invention provides an imidazo[4,5-c]quinolin-2-one compound (formula (I)), or a pharmaceutically acceptable salt thereof, that inhibits both PI3K and mTOR and, therefore, is useful in the treatment of cancer. La présente invention concerne un composé d'imidazo[4,5-c]quinolin-2-one (formula (I)), ou un sel pharmaceutiquement acceptable de celui-ci, qui inhibe à la fois PI3K et mTOR et, par conséquent, qui est utile dans le traitement du cancer.