NOVEL PROCESS FOR THE PREPARATION OF ASENAPINE

The present invention is directed to novel compounds of formula (I) as well as to the process for their preparation. Novel compounds of formula (I) can be converted into asenapine through an efficient process. The invention also relates to novel intermediates used in this process and their use in th...

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Bibliographische Detailangaben
Hauptverfasser: PEIRATS MASIA, JORDI, DALMASES BARJOAN, PERE, HUGUET CLOTET, JUAN
Format: Patent
Sprache:eng ; fre
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Beschreibung
Zusammenfassung:The present invention is directed to novel compounds of formula (I) as well as to the process for their preparation. Novel compounds of formula (I) can be converted into asenapine through an efficient process. The invention also relates to novel intermediates used in this process and their use in the preparation of compounds of formula (I). La présente invention concerne de nouveaux composés de formule I ainsi que leur procédé de synthèse. Les nouveaux composés de formule I peuvent être convertis en asénapine via un procédé efficace. La présente invention concerne également de nouveaux intermédiaires utilisés dans ce procédé et leur utilisation dans la synthèse de composés de formule I.