PROCESS FOR PREPARING BENZIMIDAZOLE COMPOUNDS

PROCESS FOR PREPARING BENZIMIDAZOLE COMPOUNDS

Provided are methods for the synthesis of heterocyclic compounds such as benzimidazole carboxylic acid core structures having Formula Ia-1 and their synthetic intermediates: wherein Z, X1, X2, X5, R2 and R10 are as defined herein. Compounds of Formula Ia-1 and their synthetic intermediates can be us...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: DEMATTEI, JOHN, FORD, JAMES GAIR, LILLEY, TIMOTHY JOHN, PISCOPIO, ANTHONY D, HACHE, BRUNO P, POINTON, SIMON MARK, LEONARD, JOHN, SHAKYA, SAGAR, PEETERS, KOEN, EVANS, MATTHEW CHARLES
Format: Patent
Sprache:eng ; fre
Schlagworte:
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
Beschreibung
Zusammenfassung:Provided are methods for the synthesis of heterocyclic compounds such as benzimidazole carboxylic acid core structures having Formula Ia-1 and their synthetic intermediates: wherein Z, X1, X2, X5, R2 and R10 are as defined herein. Compounds of Formula Ia-1 and their synthetic intermediates can be used to prepare heterocyclic derivatives such as benzimidazole derivatives. Procédés pour la synthèse de composés hétérocycliques du type structures centrales d'acide benzimidazole-carboxylique de formule Ia-1 et leurs intermédiaires synthétiques, sachant que Z, X1, X2, X5, R2 et R10 sont tels que définis dans la description. Les composés et intermédiaires décrits peuvent être utilisés pour l'élaboration de dérivés hétérocycliques du type dérivés benzimidazole.