AMPA ANTAGONISTS AND A METHOD OF TREATMENT THEREWITH
The present patent application discloses compounds having the formula or a pharmaceutically acceptable salt thereof wherein R1 is hydrogen, alkyl or benzyl; X is O or NOR2, wherein R2 is hydrogen, alkyl or benzyl; Y is N-R4 wherein R4 is hydrogen, OH or alkyl; n is 0 or 1; R6 is phenyl, naphthyl, th...
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| creator | WATJEN, FRANK DREJER, JORGEN |
| description | The present patent application discloses compounds having the formula or a pharmaceutically acceptable salt thereof wherein R1 is hydrogen, alkyl or benzyl; X is O or NOR2, wherein R2 is hydrogen, alkyl or benzyl; Y is N-R4 wherein R4 is hydrogen, OH or alkyl; n is 0 or 1; R6 is phenyl, naphthyl, thienyl, pyridyl, all of which may be substituted one or more times with substituents selected from the group consisting or halogen, CF3, NO2, amino, alkyl, alkoxy and phenyl; A is a ring of five to seven atoms fused with the benzo ring at the position s marked a and b. The compounds are useful in the treatment of cerebrovascular disorders f or example. |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | AMPA ANTAGONISTS AND A METHOD OF TREATMENT THEREWITH |
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