A PHYSICAL FORM OF N-[4-[5-(CYCLOPENTYLOXYCARBONY)AMINO-1-METHYLINDOL-3YL-METHY1]-3-METHOXYBENZOY1]-2-METHLBENZENESULPHONAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS CONTAINING IT
The invention provides a pharmaceutical composition comprising a particular physical form of N-[4-[5-(cyclopentyloxy- carbonyl)amino-1-methylindol-3-yl-methyl]-3-methoxybenzoyl]-2-methyl- benzenesulphonamide and polyvinylpyrrolidone. It also provides methods for preparing this physical form, and ano...
Gespeichert in:
Hauptverfasser: | , , , , |
---|---|
Format: | Patent |
Sprache: | eng ; fre |
Schlagworte: | |
Online-Zugang: | Volltext bestellen |
Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
container_end_page | |
---|---|
container_issue | |
container_start_page | |
container_title | |
container_volume | |
creator | TIMKO, ROBERT J HOLOHAN, JAMES J CLEMENTS, ARLENE BRADWAY, RANDY J EDWARDS, IEUAN J |
description | The invention provides a pharmaceutical composition comprising a particular physical form of N-[4-[5-(cyclopentyloxy- carbonyl)amino-1-methylindol-3-yl-methyl]-3-methoxybenzoyl]-2-methyl- benzenesulphonamide and polyvinylpyrrolidone. It also provides methods for preparing this physical form, and another physical form of N-[4-[S-(cyclopentyloxycarbonyl)amino-1-methylindol-3-yl-methyl]- -3-methoxybenzoyl]-2-methylbenzenesulphonamide useful in the preparation of the first mentioned physical form. The compositions are useful in the treatment of diseases in which leukotrienes are implicated, for example asthma. |
format | Patent |
fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_CA2056066C</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>CA2056066C</sourcerecordid><originalsourceid>FETCH-epo_espacenet_CA2056066C3</originalsourceid><addsrcrecordid>eNqFjcFqAjEQhvfiodQ-Q3O0YEDduvdxdrYbyM6ETQqmUkQknqQV7OP5cGatd08z38c_8z8VF1Cujd4gWNVI3ylpFOvNu94s9QQjWnHEIVpZR4R-JRzfoDMseq47Cm20hmuxuoz2n-ffurxt-WBF_CWDWdyMHZiY_Kd1rXB-U9NUuV6QvCc_1CsTfDbkoIdghBVwrVA6J94M7DNwAMOGP3J2XIwOu-M5vdznc_HaUMBWp9PvNp1Pu336SX9bhMVsWc2qCsvHiSu5nUyQ</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>A PHYSICAL FORM OF N-[4-[5-(CYCLOPENTYLOXYCARBONY)AMINO-1-METHYLINDOL-3YL-METHY1]-3-METHOXYBENZOY1]-2-METHLBENZENESULPHONAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS CONTAINING IT</title><source>esp@cenet</source><creator>TIMKO, ROBERT J ; HOLOHAN, JAMES J ; CLEMENTS, ARLENE ; BRADWAY, RANDY J ; EDWARDS, IEUAN J</creator><creatorcontrib>TIMKO, ROBERT J ; HOLOHAN, JAMES J ; CLEMENTS, ARLENE ; BRADWAY, RANDY J ; EDWARDS, IEUAN J</creatorcontrib><description>The invention provides a pharmaceutical composition comprising a particular physical form of N-[4-[5-(cyclopentyloxy- carbonyl)amino-1-methylindol-3-yl-methyl]-3-methoxybenzoyl]-2-methyl- benzenesulphonamide and polyvinylpyrrolidone. It also provides methods for preparing this physical form, and another physical form of N-[4-[S-(cyclopentyloxycarbonyl)amino-1-methylindol-3-yl-methyl]- -3-methoxybenzoyl]-2-methylbenzenesulphonamide useful in the preparation of the first mentioned physical form. The compositions are useful in the treatment of diseases in which leukotrienes are implicated, for example asthma.</description><edition>5</edition><language>eng ; fre</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2002</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20020402&DB=EPODOC&CC=CA&NR=2056066C$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76290</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20020402&DB=EPODOC&CC=CA&NR=2056066C$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>TIMKO, ROBERT J</creatorcontrib><creatorcontrib>HOLOHAN, JAMES J</creatorcontrib><creatorcontrib>CLEMENTS, ARLENE</creatorcontrib><creatorcontrib>BRADWAY, RANDY J</creatorcontrib><creatorcontrib>EDWARDS, IEUAN J</creatorcontrib><title>A PHYSICAL FORM OF N-[4-[5-(CYCLOPENTYLOXYCARBONY)AMINO-1-METHYLINDOL-3YL-METHY1]-3-METHOXYBENZOY1]-2-METHLBENZENESULPHONAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS CONTAINING IT</title><description>The invention provides a pharmaceutical composition comprising a particular physical form of N-[4-[5-(cyclopentyloxy- carbonyl)amino-1-methylindol-3-yl-methyl]-3-methoxybenzoyl]-2-methyl- benzenesulphonamide and polyvinylpyrrolidone. It also provides methods for preparing this physical form, and another physical form of N-[4-[S-(cyclopentyloxycarbonyl)amino-1-methylindol-3-yl-methyl]- -3-methoxybenzoyl]-2-methylbenzenesulphonamide useful in the preparation of the first mentioned physical form. The compositions are useful in the treatment of diseases in which leukotrienes are implicated, for example asthma.</description><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2002</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqFjcFqAjEQhvfiodQ-Q3O0YEDduvdxdrYbyM6ETQqmUkQknqQV7OP5cGatd08z38c_8z8VF1Cujd4gWNVI3ylpFOvNu94s9QQjWnHEIVpZR4R-JRzfoDMseq47Cm20hmuxuoz2n-ffurxt-WBF_CWDWdyMHZiY_Kd1rXB-U9NUuV6QvCc_1CsTfDbkoIdghBVwrVA6J94M7DNwAMOGP3J2XIwOu-M5vdznc_HaUMBWp9PvNp1Pu336SX9bhMVsWc2qCsvHiSu5nUyQ</recordid><startdate>20020402</startdate><enddate>20020402</enddate><creator>TIMKO, ROBERT J</creator><creator>HOLOHAN, JAMES J</creator><creator>CLEMENTS, ARLENE</creator><creator>BRADWAY, RANDY J</creator><creator>EDWARDS, IEUAN J</creator><scope>EVB</scope></search><sort><creationdate>20020402</creationdate><title>A PHYSICAL FORM OF N-[4-[5-(CYCLOPENTYLOXYCARBONY)AMINO-1-METHYLINDOL-3YL-METHY1]-3-METHOXYBENZOY1]-2-METHLBENZENESULPHONAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS CONTAINING IT</title><author>TIMKO, ROBERT J ; HOLOHAN, JAMES J ; CLEMENTS, ARLENE ; BRADWAY, RANDY J ; EDWARDS, IEUAN J</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_CA2056066C3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2002</creationdate><topic>ACYCLIC OR CARBOCYCLIC COMPOUNDS</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>TIMKO, ROBERT J</creatorcontrib><creatorcontrib>HOLOHAN, JAMES J</creatorcontrib><creatorcontrib>CLEMENTS, ARLENE</creatorcontrib><creatorcontrib>BRADWAY, RANDY J</creatorcontrib><creatorcontrib>EDWARDS, IEUAN J</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>TIMKO, ROBERT J</au><au>HOLOHAN, JAMES J</au><au>CLEMENTS, ARLENE</au><au>BRADWAY, RANDY J</au><au>EDWARDS, IEUAN J</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>A PHYSICAL FORM OF N-[4-[5-(CYCLOPENTYLOXYCARBONY)AMINO-1-METHYLINDOL-3YL-METHY1]-3-METHOXYBENZOY1]-2-METHLBENZENESULPHONAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS CONTAINING IT</title><date>2002-04-02</date><risdate>2002</risdate><abstract>The invention provides a pharmaceutical composition comprising a particular physical form of N-[4-[5-(cyclopentyloxy- carbonyl)amino-1-methylindol-3-yl-methyl]-3-methoxybenzoyl]-2-methyl- benzenesulphonamide and polyvinylpyrrolidone. It also provides methods for preparing this physical form, and another physical form of N-[4-[S-(cyclopentyloxycarbonyl)amino-1-methylindol-3-yl-methyl]- -3-methoxybenzoyl]-2-methylbenzenesulphonamide useful in the preparation of the first mentioned physical form. The compositions are useful in the treatment of diseases in which leukotrienes are implicated, for example asthma.</abstract><edition>5</edition><oa>free_for_read</oa></addata></record> |
fulltext | fulltext_linktorsrc |
identifier | |
ispartof | |
issn | |
language | eng ; fre |
recordid | cdi_epo_espacenet_CA2056066C |
source | esp@cenet |
subjects | ACYCLIC OR CARBOCYCLIC COMPOUNDS CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
title | A PHYSICAL FORM OF N-[4-[5-(CYCLOPENTYLOXYCARBONY)AMINO-1-METHYLINDOL-3YL-METHY1]-3-METHOXYBENZOY1]-2-METHLBENZENESULPHONAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS CONTAINING IT |
url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-03T10%3A51%3A10IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=TIMKO,%20ROBERT%20J&rft.date=2002-04-02&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3ECA2056066C%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |