MEDICAMENTS
The use of a compound of formula I (I) wherein R is a hydrogen atom or a group selected from Cl 6alkyl (optionally substituted by C3-7cycloalkyl), C3-6 alkenyl, C3-6alkynyl, C3-7 cycloalkyl, aralkyl (in which the alkyl moiety contains 1-5 carbon atoms) and -CHO; R1 and R2, which may be the same or d...
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Zusammenfassung: | The use of a compound of formula I (I) wherein R is a hydrogen atom or a group selected from Cl 6alkyl (optionally substituted by C3-7cycloalkyl), C3-6 alkenyl, C3-6alkynyl, C3-7 cycloalkyl, aralkyl (in which the alkyl moiety contains 1-5 carbon atoms) and -CHO; R1 and R2, which may be the same or different, represent a hydrogen atom, a halogen atom or a group selected from C1-4alkyl, C1-4alkoxy, hydroxyl, cyano, nitro and -NR3R4 where R3 and R4 is each a hydrogen atom or a C1-4alkyl group and X is an oxygen atom or a group -CH2; or a physiologically acceptable salt or hydrate thereof for treating, relieving or preventing the effects of sexual dysfunction. Preferred compounds include trans-5-fluoro-2,3,3a,9a-tetrahydro-lH-1,4! benzodioxino 2,3-clpyrrole and trans-5-fluoro-1,2,3,3a,9,9a-hexahydro1! benzopyrano 2,3-c!pyrrole. Conditions that may be treated in this manner include, in the case of the male, erectile inadequacy and, in the case of the female, sexual arousal disorder. AD120/
The use of a compound of formula I (I) wherein R is a hydrogen atom or a group selected from Cl 6alkyl (optionally substituted by C3-7cycloalkyl), C3-6 alkenyl, C3-6alkynyl, C3-7 cycloalkyl, aralkyl (in which the alkyl moiety contains 1-5 carbon atoms) and -CHO; R1 and R2, which may be the same or different, represent a hydrogen atom, a halogen atom or a group selected from C1-4alkyl, C1-4alkoxy, hydroxyl, cyano, nitro and -NR3R4 where R3 and R4 is each a hydrogen atom or a C1-4alkyl group and X is an oxygen atom or a group -CH2; or a physiologically acceptable salt or hydrate thereof for treating, relieving or preventing the effects of sexual dysfunction. Preferred compounds include trans-5-fluoro-2,3,3a,9a-tetrahydro-lH-¢1,4! benzodioxino ¢2,3-clpyrrole and trans-5-fluoro-1,2,3,3a,9,9a-hexahydro¢1! benzopyrano ¢2,3-c!pyrrole. Conditions that may be treated in this manner include, in the case of the male, erectile inadequacy and, in the case of the female, sexual arousal disorder. AD120/ |
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