PROCESS FOR THE PREPARATION OF A THIAZEPINE COMPOUND

11-(4-¢2-(2-Hydroxyethoxy)ethyl!-piperazinyl)-dibenzo¢b,f!¢1,4!thiazepine and the salts thereof possess antiandropaninergic activity, especially antipyschotic activity, and are prepared by reacting 11-piperazinyldibenzo¢b,f!¢1,4!thiazepine with a compound of the formula: X-CH2-CH2-O-CH2-CH2OH (where...

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Bibliographische Detailangaben
Hauptverfasser: COPELAND, ROBERT JEFFREY, BARKER, ALAN CHARLES
Format: Patent
Sprache:eng ; fre
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Zusammenfassung:11-(4-¢2-(2-Hydroxyethoxy)ethyl!-piperazinyl)-dibenzo¢b,f!¢1,4!thiazepine and the salts thereof possess antiandropaninergic activity, especially antipyschotic activity, and are prepared by reacting 11-piperazinyldibenzo¢b,f!¢1,4!thiazepine with a compound of the formula: X-CH2-CH2-O-CH2-CH2OH (wherein X represent an atom or group removable as an anion and, where appropriate further reaction of the product obtained to yield the free base or salt as desired.