VERFAHREN ZUR HERSTELLUNG VON ASPARTYL- CYCLOHEXYLALANINAMID
Disclosure is a method for preparing alpha-aspartyl-beta-cyclohexylalaninamide, comprising carrying out a first step of amide formation of an alpha-aspartyl phenylamine ester of general formula (II)wherein: R is a C1-C4 alkyl radical, and then performing a catalytic hydrogenation of the resulting al...
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| Zusammenfassung: | Disclosure is a method for preparing alpha-aspartyl-beta-cyclohexylalaninamide, comprising carrying out a first step of amide formation of an alpha-aspartyl phenylamine ester of general formula (II)wherein: R is a C1-C4 alkyl radical, and then performing a catalytic hydrogenation of the resulting alpha-aspartyl phenylalaninamide ammonium salt, optionally released previously from its salt, and optionally transforming it into an addition acis salt. |
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