A Practical One-Pot Synthesis of 5-Aryl-2-furaldehydes

Abstract A useful one-pot synthesis of 5-aryl-2-furaldehydes via palladium-mediated Suzuki coupling of aryl halides with in situ generated 5-(diethoxymethyl)-2-furylboronic acid is described. The procedure has general applicability, delivers high yields, and is amenable to scale-up.

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Bibliographische Detailangaben
Veröffentlicht in:	Synthesis (Stuttgart) 2001, Vol.2001 (11), p.1681-1685
Hauptverfasser:	McClure, Michael S., Roschangar, Frank, Hodson, Stephen J., Millar, Alan, Osterhout, Martin H.
Format:	Artikel
Sprache:	eng
Online-Zugang:	Volltext
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Beschreibung
Zusammenfassung:	Abstract A useful one-pot synthesis of 5-aryl-2-furaldehydes via palladium-mediated Suzuki coupling of aryl halides with in situ generated 5-(diethoxymethyl)-2-furylboronic acid is described. The procedure has general applicability, delivers high yields, and is amenable to scale-up.
ISSN:	0039-7881 1437-210X
DOI:	10.1055/s-2001-16759