Synthesis of 2-Arylpyrazolo[1,5-a]pyridines by Suzuki–Miyaura Cross-Coupling Reaction
Abstract Convenient access to a variety of 2-arylated pyrazolo[1,5- a ]pyridine via pyrazolo[1,5- a ]pyridine-2-yl triflate using the Suzuki–Miyaura cross-coupling reaction is described. Fifteen 2-arylpyrazolo[1,5- a ]pyridine derivatives were synthesized in 52–95% yields.
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| Veröffentlicht in: | Synthesis (Stuttgart) 2015-10, Vol.47 (20), p.3221-3230 |
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| Hauptverfasser: | , , , , |
| Format: | Artikel |
| Sprache: | eng |
| Online-Zugang: | Volltext |
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| Zusammenfassung: | Abstract
Convenient access to a variety of 2-arylated pyrazolo[1,5-
a
]pyridine via pyrazolo[1,5-
a
]pyridine-2-yl triflate using the Suzuki–Miyaura cross-coupling reaction is described. Fifteen 2-arylpyrazolo[1,5-
a
]pyridine derivatives were synthesized in 52–95% yields. |
|---|---|
| ISSN: | 0039-7881 1437-210X |
| DOI: | 10.1055/s-0034-1381025 |