Copper acetate - Iodine co-mediated thiolation of 2-arylpyridines with thiophenol

Copper acetate - iodine co-mediated regioselective ortho-arylthiolation of 2-arylpyridines has been accomplished with inexpensive and convenient thiophenol as the arylthiolating reagent. This protocol features excellent functional group tolerance, generating thioarylated products in moderate-to-high...

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Veröffentlicht in:	Tetrahedron 2022-01, Vol.103, p.132552, Article 132552
Hauptverfasser:	He, Yayun, Hou, Senpeng, Hu, Junhao
Format:	Artikel
Sprache:	eng
Schlagworte:	2-arylpyridines Copper acetate Orthoarylthiolation Thiophenol
Online-Zugang:	Volltext
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Beschreibung
Zusammenfassung:	Copper acetate - iodine co-mediated regioselective ortho-arylthiolation of 2-arylpyridines has been accomplished with inexpensive and convenient thiophenol as the arylthiolating reagent. This protocol features excellent functional group tolerance, generating thioarylated products in moderate-to-high yields. © 2021 Elsevier Science. All rights reserved. [Display omitted]
ISSN:	0040-4020 1464-5416
DOI:	10.1016/j.tet.2021.132552