ChemInform Abstract: Catalytic Enantioselective Synthesis of α-Arylaminocyclobutanones

Optimized conditions allow the enantioselective synthesis of the title compounds from racemic α‐hydroxycyclobutanone and N‐alkylaniline derivatives via a tandem condensation/keto‐enol tautomerization process.

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Bibliographische Detailangaben
Veröffentlicht in:	ChemInform 2014-09, Vol.45 (35), p.no-no
Hauptverfasser:	Aitken, David J., Caboni, Pierluigi, Eijsberg, Hendrik, Frongia, Angelo, Guillot, Regis, Ollivier, Jean, Piras, Pier Paolo, Secci, Francesco
Format:	Artikel
Sprache:	eng
Schlagworte:	amination amination, N‐alkylation, N‐arylation amines (benzene compounds) catalysis catalysis, phase‐transfer catalysis cyclobutane derivatives N-alkylation N-arylation phase-transfer catalysis
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Beschreibung
Zusammenfassung:	Optimized conditions allow the enantioselective synthesis of the title compounds from racemic α‐hydroxycyclobutanone and N‐alkylaniline derivatives via a tandem condensation/keto‐enol tautomerization process.
ISSN:	0931-7597 1522-2667
DOI:	10.1002/chin.201435076