Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990

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Veröffentlicht: Oxford [u.a.] Pergamon Press 1991
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Schriftenreihe:Advances in the biosciences 82
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adam_text IMAGE 1 CONTENTS PREFACE XIX PHYSIOLOGICAL AND PHARMACOLOGICAL RELEVANCE OF PRESYNAPTIC RECEPTORS IN NEUROTRANSMISSION S.Z. LANGER, I. ANGEL AND H. SCHOEMAKER 1 PRE- AND POSTJUNCTIONAL MUSCARINIC RECEPTORS IN THE GUINEA-PIG TRACHEA H. KILBINGER, D. WOLF AND G. D AGOSTINO 7 PRESYNAPTIC A-AUTOADRENOCEPTORS ON PERIPHERAL NORADRENERGIC NEURONES OF NEWBORN RABBITS AND DOGS S. GUIMARAES, M.Q. PAIVA, D. MOURA AND M J. VAZ-DA-SILVA 11 CHOLINERGIC-ADRENERGIC PRESYNAPTIC INTERACTIONS IN THE HEART AND CHARACTERIZATION OF THE RECEPTORS INVOLVED E. MUSCHOLL, A. HABERMEIER-MUTH, U. ALTES AND K. FORSYTH 15 STRUCTURAL REQUIREMENTS FOR DA2 (PERIPHERAL) DOPAMINE RECEPTOR AGONIST ACTIVITY J.D. KOHLI AND P.T. HORN 19 A2-ADRENOCEPTOR MODULATION OR NORADRENALINE RELEASE IN HUMAN AND RABBIT RENAL ARTERIES: CLONIDINE ACTS AS A PARTIAL AGONIST L.C. RUMP, G. RUFF AND P. SCHOLLMEYER 23 EFFECT OF A2-ADRENOCEPTOR ANTAGONISTS ON NOREPHINE RELEASE AND INHIBITION OF INSULIN SECRETION DURING PANCREATIC NERVE STIMMULATION. INTERACTIONS AT PRE- AND POSTSYNAPTIC SITES N. DUVAL, I. ANGEL, A. OBLIN, M.T. EON AND S.Z. LANGER 25 IMAGE 2 VI CONTENTS ANTAGONIST ACTIVITY OF SL 84.0418 AND IDAZOXAN AT PRE AND POST SYNAPTIC 2-ADRENORECEPTORS H. SHOEMAKER, A. GROSSET, I. ANGEL AND S.Z. LANGER 27 DOES THE DISTANCE BETWEEN NERVE VARICOSITIES AND ADRENOCEPTORS PLAY ANY ROLE IN THE RELATIVE CONTRIBUTION OF ATP/NORADRENALINE FOR POSTJUNCTIONAL RESPONSE? J. GONGALVES, F. CARVALHO AND S. GUIMARAES 29 IN VIVO PRESYNAPTIC INTERACTION BETWEEN 5-HT AND ADRENERGIC ANTAGONISTS ON NORADRENERGIC NEUROTRANSMISSION M. DAVY, F. BESLOT, M. MIDOL-MONNET, M. HEIMBURGER & Y. COHEN 31 ACTIVITY OF N-ETHYL-NOR-ARECAIDINE PROPARGYL ESTER AND (R)-NIPECOTIC ACID ETHYL ESTER AT PRE-AND POSTSYNAPTIC MUSCARINIC RECEPTOR SUBTYPES M. ELTZE, F. DORJE, H. TIETZ, A. IMMEL, E. MUTSCHLER AND G. LAMBRECHT 33 EFFECTS OF NEUROMUSCULAR BLOCKING AGENTS ON NEURONAL NICOTINE RECEPTORS OF MOTOR NERVES: BLOCKADE OF NICOTINIC AUTOFACILITATION AND BACKFIRING I. WESSLER, E. JUNG, K. WAGENMANN, T. VOGT AND R. BESSER 35 A RAPID IN VITRO ASSAY OF THE HISTAINE H3-RECEPTOR: INHIBITION OF ELECTRICALLY EVOKED CONTRACTIONS OF GUINEA- PIG ILEUM PREPARATIONS G J. MENKVELD AND H. TIMMERMAN 37 FACTORS INFLUENCING THE FUNCTION OF PRESYNAPTIC A2-ADRENOCEPTORS IN RAT BRAIN P J. HOLLINGSWORTH AND C.B. SMITH 39 PRESYNAPTIC DOPAMINERGIC AUTORECEPTORS AS TARGETS FOR DRUGS A. CARLSSON 43 IMAGE 3 CONTENTS VII DOPA ITSELF FACILITATES NORADRENALINE RELEASE VIA PRESYNAPTIC FL-ADRENOCEPTORS IN RAT HYPOTHALAMIC SLICES - DOPA IS PROBABLY A NEUROACTIVE SUBSTANCE Y. MISU, Y. GOSHIMA AND S. NAKAMURA 47 THE THIRD DOPAMINE RECEPTOPR (D3) AS AN AUTORECEPTOR J.C.SCHWARTZ, P. SOKOLOFF, B. GIROS, M.P. MARTRES AND M.L. BOUTHENET 51 TERMINAL DOPAMINERGIC AUTORECEPTORS ARE OF MINOR IMPORTANCE FOR THE SEDATION PRODUCED BY DA RECEPTOR AGONISTS IN RATS S. AHLENIUS, V. HILLEGAART AND L. SVENSSON 55 MODULATION OF 5-HT RELEASE BY PRESYNAPTIC INHIBITORY AND FACILITATORY 5-HT RECEPTORS IN BRAIN SLICES A.M. GALZIN AND S.Z. LANGER 59 MODULATION OF 5-HYDROXYTRYPTAMINE AND NORADRENALINE RELEASE IN THE BRAIN AND RETINA VIA PRESYNAPTIC HETERORECEPTORS: SOME NEW ASPECTS M. GOTHERT, E. SCHLICKER, K. FINK AND G. MOLDERINGS 63 AUTORECEPTORS AND HETERORECEPTORS EVIDENCED BY HISTAMINE H3 RECEPTOR LIGANDS M. GARBARG, J.M. ARRANG, C. LLORENS-CORTES, H. POLLARD, A. ROULEAU, J.C. SCHWARTZ, M.D. TRUNG TUONG, R. LIPP, H. STARK, W. SCHUNACK AND J.M. J^ECOMTE 67 SOMATO-DENDRITIC 5-HTIA AUTORECEPTORS IN THE DORSAL RAPHE NUCLEUS; PHARMACOLOGICAL AND FUNCTIONAL PROPERTIES M. HAMON, S. EL MESTIKAWY, L. LANFUMEY, J. ADRIEN, C.M. FATTACCINI AND H. GOZLAN 71 AUTORECEPTOR-MEDIATED CONTROL OF SEROTONIN RELEASE IN THE RAT BRAIN IN VIVO B SCATTON, L. ROUQUIER, G. BONVENTO, A. SERRANO AND P. BLIER 75 IMAGE 4 VIII CONTENTS EFFECTS OF A2-ADRENOCEPTOR AGONIST AND ANTAGONIST ON SPATIAL MEMORY IN RATS M.M. AIRAKSINEN, S.A. NIEMINEN, E.J. MACDONALD, J. SIRVIO AND P.J. RIEKKINEN, JR. 79 MODULATION OF THE CA 2+ -EVOKED RELEASE OF DOPAMINE FROM SYNAPTOSOMES N. WEINER, J.F. BOWYER AND J. MASSERANO 81 EVIDENCE AGAINST A DIRECT LINK BETWEEN SEROTONIN UPTAKE SITES AND PRESYNAPTIC SEROTONIN AUTORECEPTORS N. LIMBERGER, E. SINGER AND K. STARKE 85 A COMPARISON OF PRESYNAPTIC SEROTONIN AUTORECEPTORS IN RABBIT, RAT AND GUINEA-PIG BRAIN CORTEX R. DEICHER, N. LIMBERGER AND K. STARKE 87 SEROTONERGIC MODULATION OF THE RELEASE OF [ 3 H] GABA FROM GUINEA-PIG HIPPOCAMPAL SYNAPTOSOMES I. CLOEZ, C. HAREL-DUPAS AND G. FILLION 89 PRE- AND POST-SYNAPTIC LOCATION OF 5-HT 3 RECEPTORS IN THE RAT SPINAL CORD A.M. LAPORTE, M.C. LOMBARD, S. BOURGOIN, D. VERGE, H. GOZLAN AND M. HAMON 91 DISTRIBUTION OF [ 3 H]SCH 23390 BINDING SITES IN THE HUMAN SUBSTANTIA NIGRA F. THIBAUT, E.C. HIRSCH, R. RAISMAN, F. JAVOY-AGID AND Y. AGID 93 PRESYNAPTIC REGULATION OF DOPAMINE RELEASE FROM SYNAPTOSOMES OF THE RAT STRIATUM IS CONTROLLED BY DIFFERENT TYPES OF GLUTAMATE RECEPTORS J.M. DESCE, G. GODEHEU, A. CHERAMY AND J. GLOWINSKI 95 MICRODIALYSIS STUDIES OF THE EFFECTS OF LOCAL APOMORPHINE INFUSIONS ON DOPAMINE RELEASE IN RAT STRIATUM M. GOINY, T. GUIX, M. HERRERA-MARSCHITZ AND U. UNGERSTEDT 97 IMAGE 5 CONTENTS IX DOPAMINERGIC HETERO-REGULATION OF STRIATAL FT-OPIATE RECEPTORS: FURTHER EVIDENCE FOR THEIR POSTSYNAPTIC LOCATION F. TROVERO, D. HERVE, M. DESBAN, J. GLOWINSKI AND J.P. TASSIN 99 PRESYNAPTIC MODULATION OF STRIATAL DOPAMINE RELEASE BY ENKEPHALINS N. DOURMAP, A. MICHAEL-TITUS AND J. COSTENTIN 101 MODULATION OF DOPAMINE AND ACETYLCHOLINE RELEASE IN THE RABBIT CAUDATE NUCLEUS BY OPIOIDS: RECEPTOR TYPE AND INTERACTION WITH AUTORECEPTORS R. JACKISCH, H. HOTZ AND G. HERTTING 103 PRESYNAPTIC AUTORECEPTORS MAY CONTROL THE RELEASE OF MET- ENKEPHALIN FROM THE RAT SPINAL CORD E. COLLIN, S. BOURGOIN, D. CHANTREL, J J. BENOLIEL, A. MAUBORGNE, M. HAMON AND F. CESSELIN 105 INVOLVEMENT OF NMDA RECEPTORS IN THE PRESYNAPTIC REGULATION OF DOPAMINE RELEASE IN STRIOSOME- AND MATRIX-ENRICHED AREAS OF THE RAT STRIATUM M.-O. KREBS, M.-L. KERNEL, M. DESBAN, J. GLOWINSKI AND C. GAUCHY 107 INHIBITION OF SYNAPTOSOMAL TYROSINE HYDROXYLASE BY DOPAMINE AUTORECEPTORS: ROLE CA 2+ AND K + P. ONALI, E. MOSCA AND M.C. OLIANAS 109 DOPAMINERGIC MODULATION OF STRIATAL SENSORY RESPONSES T.I. LIDSKY, C. MANETTO AND S.P. BANERJEE 111 SELECTIVE PRESYNAPTIC DOPAMINE AGONIST TREATMENT OF SCHIZOPHRENIA WITH BHT-920 P. WINCKLER AND M. BARTELS 113 EFFECTS OF THE ANTIPARKINSONIAN DRUGS AMANTADINE AND MEMANTINE ON STRIATAL NEUROTRANSMITTER RELEASE IN VITRO A. LUPP, T. LINK, G. HERTTING, R. JACKISCH AND T J. FEUERSTEIN 117 IMAGE 6 X CONTENTS TRANSMITTER INTERACTIONS IN STRIATUM MAY OCCUR VIA EFFECTS ON HIGH AFFINITY TRANSPORTERS G. LONART, S. BERNATH AND M J. ZIGMOND 119 A COMPARISON OF THE EFFECT OF BACLOFEN ON RADIOLABELLED GABA AND NORADERNALINE RELEASE IN RAT CORTICAL SLICES C. ENNIS AND M.C.W. MINCHIN 121 EFFECTS OF CHRONIC TREATMENT WITH FLUNITRAZEPAM ON GABA A ADENOSINE AND GLUTAMATE RECEPTOR PLASTICITY IN RATS M. BARALDI, P. ZANOLI, A. GIACOBAZZI, G. VACCARI AND R. AVALLONE 123 MODULATION OF N-METHYL-D-ASPARTATE (NMDA)-STIMULATED NORADRENALINE RELEASE IN RAT BRAIN CORTEX BY PRESYNAPTIC A2-ADRENOCEPTORS AND HISTAMINE KB RECEPTORS K. FINK, E. SCHLICKER AND M. GOTHERT 125 NORADRENALINE RELEASE IN THE PIG RETINA AND ITS HISTAMINE H 3 RECEPTOR-MEDIATED INHIBITION E. SCHLICKER AND M. GOTHERT 127 STRUCTURE AND FUNCTION OF THE GABA REUPTAKE SYSTEM B.I. KANNER 129 ENERGIZING THE VACUOLAR SYSTEM OF EUKARYOTIC CELLS N. NELSON 135 THE MOLECULAR SIZE OF THE NEURONAL NORADENALINE CARRIER H. BONISH, J. MICHAEL-HEPP, B. BLUM AND G. MARTINY-BARON 139 IDENTIFICATION AND REGULATION OF HIGH-AFFINITY-CHOLINE TRANSPORTER M. KNIPPER 143 KETANSERIN AS A LIGAND OF THE VESICULAR MONOAMINE TRANSPORTER J.P. HENRY, B. GASNIER, M.F. ISAMBERT, F. DARCHEN AND D. SCHERMAN 147 IMAGE 7 CONTENTS XI DOPAMINE TRANSPORTER - COCAINE RECEPTOR: CHARACTERIZATION AND PURIFICATION R. SIMANTOV, R. VAUGHAN, R. LEW, A. WILSON AND M.J. KUHAR 151 CHARACTERIZATON AND PURIFICATION OF THE SEROTONIN TRANSPORTER LOCATED AT THE CYTOPLASMIC MEMBRANE OF HUMAN PLATELETS: A THREE-STEP STRATEGY J.M. LAUNAY, C. CHOPIN-ROBERT, C. GEOFFROY, D. BONDOUX, D. LAMBLIN, M.L. GIRON, V. MUTEL, M.H. BUC-CARON, J. LASNERET, O. KELLERMANN, D. DA PRADA AND J.E. ALOUF 155 MOLECULAR CHARACTERIZATION OF THE NEURONAL SODIUM-ION COUPLED 5-HYDROXYTRYPTAMINE TRANSPORTER D. GRAHAM, H, ESNAUD AND S.Z. LANGER 159 KINETIC ANALYSES OF THE NA + AND CL DEPENDENCES OF THE SYNAPTOSOMAL SPECIFIC UPTAKE OF 3 H DOPAMINE N. CHAB, J.-J. BONNET AND J. COSTENTIN 163 LOCALIZATION OF DOPAMINE UPTAKE COMPLEX BY BTCP ON RAT BRAIN SECTIONS AND DOPAMINERGIC NEURONS IN VITRO C. CERRUTI, J.-M. KAMENKA AND A. PRIVAT 165 IN VIVO BINDING OF [ 3 H]GBR 12783 IN MOUSE BRAIN - CHARACTERISTICS OF THE LABELLING OF STRIATAL DOPAMINE UPTAKE SITES J.-M. VAUGEOIS, J.-J. BONNET AND J. COSTENTIN 167 [ 3 H]GBR 12935 BINDS TO MEMBRANE FROM THE HUMAN PLATELET B. DEAN AND D.L. COPOLOV 169 DOPAMINE TRANSPORTER IN AGING I. SHIMIZU AND C. PRASAD 171 SODIUM DEPENDENT, HIGH AFFINITY CHOLINE TRANSPORT EXPRESSED IN OOCYTES S. O REGAN, S. BIRMAN AND F.M. MEUNIER 175 IMAGE 8 XII CONTENTS COMPARISON OF THE EFFECTS OF VESAMICOL AND OF CETIEDIL ANALOGUES ON ACETYLCHOLINE RELEASE AND VESICULAR ACETYLCHOLINE TRANSPORT M.F. DIEBLER, Y. MOROT GAUDRY-TALARMAIN, J.C. LANCELOT, M. ROBBA, J.L. MORGAT AND M. ISRAEL 177 DOPAMINE MODULATES [ 3 H]BTCP (A PHENCYCLIDINE DERIVATIVE) BINDING TO THE DOPAMINE UPTAKE COMPLEX J. VIGNON, T. MAURICE, G. BARBANEL AND J.M. KAMENKA 179 THE HETEROGENEOUS LABELLING WITH 3 H-NORADRENALINE OF THE INCUBATED VAS DEFERENS OF THE RAT U. TRENDELENBURG, C.-L. SCHONFELD, T. HALBRIIGGE AND E. SCHOMIG 181 ALTERATIONS IN PLATELET [ 3 H]-IMIPRAMINE BINDING, 5HT UPTAKE AND PLASMA A I -ACID GLYCOPROTEIN CONCENTRATIONS IN PATIENTS WITH MAJOR DEPRESSION D.L. KNIGHT, T.A. SLOTKIN, L.R. MEYERSON, K.R.R. KRISHNAN AND C.B. NEMEROFF 185 IONIC AND TEMPERATURE DEPENDENCES OF THE 3 H DOPAMINE SPECIFIC UPTAKE AND 3 H GBR 12783 OR 3 H MAZINDOL SPECIFIC BINDING ON THE DOPAMINE NEURONAL CARRIER J.-J. BONNET, S. BENMANSOUR, N. CHAB, J. COSTENTIN, E.M. PARKER AND L.X. CUBEDDU 189 DYNAMIC PROPERTIES OF MONAMINE STORAGE VESICLES: PHARMACOLOGICAL AND PHYSIOLOGICAL IMPLICATIONS C. DESNOS, F. DARCHEN, Y. MASUO, W. ROSTENE AND D. SCHERMAN 193 GAB A UPTAKE INHIBITORS: KINETICS AND MOLECULAR PHARMACOLOGY O.M. LARSSON, E. FALCH, A. SCHOUSBOE AND P. KROGSGAARD-LASEN 197 COEXISTANCE OF MORE THAN ONE NEUROTRANSITTER UPTAKE SYSTEM ON THE SAME NERVE TERMINAL IN THE BRAIN M. RAITERI, G. BONANNO, M. PENDE AND S. SETTI 201 IMAGE 9 CONTENTS XIII PEPTIDERGIC REGULATION OF STRIATAL DOPAMINE TRANSPORTER COMPLEX C. PRASAD 207 DIFFERENT INTERACTIONS OF CITALOPRAM WITH THE PREJUNCTIONAL EFFECTS OF SEROTONIN IN PERPHERAL TISSUES E. ADLER-GRASCHINSKY, N.V. BUTTA, A. B. ELGOYHEN AND P.S. LORENZO 213 EVOLUTION OF THE VESICULAR MONOAMINE TRANSPORTER DURING AGEING IN THE RAT BRAIN: A QUANTITATIVE AUTORADIOGRAPHIC STUDY WITH 3 H DIHYDROTETRABENAZINE I. LEROUX-NICOLLET AND J. COSTENTIN 219 INFLUENCE OF THE OXYGEN DISPONIBILITY ON THE EFFICIENCY OF THE NEURONAL DOPAMINE UPTAKE COMPLEX B. NAUDIN, CH.SALIGAUT AND J. COSTENTIN 221 DIFFERENCES IN BEHAVIOURAL RESPONSES ELICITED BY DEXAPHETAMINE AND THE PURE DOPAMINE UPTAKE INHIBITOR GBR 12783 D. DUTERTE-BOUCHER AND J. COSTENTIN 223 PROTECTION OF THE SYNAPTOSOMAL 5-HT UPTAKE SYSTEM BY A GINKGO BILOBA EXTRACT (GBE 761) C. RAMASSAMY AND J. COSTENTIN 225 THE BINDING OF NORADENALINE TO THE SUBSTRATE RECOGNITION SITE OF THE NEURONAL NORADRENALINE CARRIER (UPTAKEI) DEPENDS ON SODIUM AND CHLORIDE E. SCHOMIG 227 IN VIVO DISTRIBUTION OF RADIOLABELLED CITALOPRAM IN BRAIN AS A MARKER OF 5-HT UPTAKE SITES FOR PET S.P. HUME, J.E. CREMER, V.W. PIKE, C. PASCALI, A.A. LAMMERTSMA, R. DOLAN AND C.J. BENCH 229 RELATIONSHIP OF [ 3 H] PAROXETINE BINDING AND 5-HT RECOGNITION SITES ON THE NEURONAL SEROTONIN TRANSPORTER B. FOY, A. HEPNER AND P.D. HRDINA 231 IMAGE 10 XIV CONTENTS EFFECTS OF REPEATED ADMINISTRATION OF ANTIDEPRESSANTS ON SEROTONIN UPTAKE SITES MEASURED USING [ 3 H] CYANOIMIPRAMINE AUTORADIOGRAPHY D J. BRUNSWICK, G.B. KOVACHICH, C.E. ARONSON AND A. FRASER 233 RAPID CHANGES IN 3 H-IMIPRAMINE BINDING IN PLATELETS OF DEPRESSED PATIENTS AFTER AMINEPTINE TREATMENT R. JEANNINGROS, B. GRONIER, J.M. AZORIN AND R. TISSOT 235 BRAIN 5-HT UPTAKE SITES, LABELLED WITH [ 3 H]PAROXETINE, IN DEPRESSED SUICIDES K.M. LAWRENCE, F. DE PAERMENTIER, S.C. CHEETHAM, M.R. CROMPTON, C.L.E. KATONA AND R.W. HORTON 237 PINOLINE, THE NATURAL LIGAND OF SEROTONIN TRANSPORTER IN RETINA AND PINEAL GLAND M.M. AIRAKSINEN AND E. KARI 239 DIFFERENTIAL INTERACTION OF PHENCYCLIDINE (PCP) WITH THE DOPAMINE UPTAKE COMPLEX AND THE PCP RECEPTOR IN VIVO T. MAURICE, J. VIGNON, J.-M. KAMENKA, J.-L. PIRAT AND R. CHICHEPORTICHE 241 THE UPTAKE OF THE AMINO ACID L-ALANINE ON ITS INHIBITORY PRESYNAPTIC EFFECTS IN RAT ISOLATED ATRIA N.V. BUTTA, D.S. HANSEN AND E. ADLER-GRASCHINSKY 243 ROLE OF OMEGA (BZD) SITES OF THE G A B AA RECEPTOR MACROMOLECULAR COMPLEX IN THE MODULATION OF SEROTONIN RELEASE A. LISTA, S. ARBILLA AND S.Z. LANGER 245 MECHANISMS OF INHIBITION OF TRANSMITTER RELEASE BY ADENOSINE ANALOGS B.B. FREDHOLM, P.-S. HU, I. VAN DER PLOEG, M. DUNER-ENGSTROM AND T.V. DUNWIDDIE 249 IMAGE 11 261 CONTENTS XV DEPENDENCE OF THE AI-ADENOSINE RECEPTOR-MEDIATED INHIBITION OF [ 3 H] NORADRENALINE RELEASE IN HIPPOCAMPUS ON THE STIMULATION CONDITIONS C. ALLGAIER, R. GREBER, M. HIPPACH AND G. HERTTING 253 MODULATION OF [ 3 H]-SEROTONIN RELEASE IN RAT SPINAL CORD SYNAPTOSOME VIA DIHYDROPYRIDINE-SENSITIVE CALCIUM CHANNELS AND PROTEIN KINASE C D J. JONES AND V.C. GANDHI 257 G-PROTEINS AND PREJUNCTIONAL A-ADRENOCEPTORS T.V. MURPHY AND H. MAJEWSKI OPIOID INHIBITION OF OXYTOCIN RELEASE, BUT NOT AUTOINHIBITION OF DOPAMINE RELEASE MAY INVOLVE ACTIVATION OF POTASSIUM (K + ) CHANNELS K RACK6, U. HAAS, S. SPERB, A. FISCHBACH, H. HOF, S. SIRRENBERG AND R. WAMMACK 265 3,4-DIAMINOPYRIDINE-EVOKED NORADRENALINE RELEASE IN HIPPOCAMPAL SLICES: FURTHER PROPERTIES AND INVOLVEMENT OF ADENYLATE CYCLASE R. JACKISCH, H. RENSING, H.Y. HUANG, C. ALLGAIER AND G. HERTTING 269 INTERNEURONAL CYCLIC GMP AND EDRF-LIFE SUBSTANCE MODULATE NOREPINEPHRINE RELEASE FROM PERIPHERAL SYMPATHETIC NERVES S. GREENBERG, F . P J. DIECKE, M. WANG, J. XIE AND T.P. TANAKA 271 MODULATORY ROLE OF NEUROPEPTIDE Y AND PEPTIDE YY AT THE NMDA RECEPTOR COMPLEX F J. ROMAN, X. PASCAUD, O. DUFFY AND J.L. JUNIEN 275 PREJUNCTIONAL NEUROPEPTIDE Y RECEPTORS ARE LINKED TO A G-PROTEIN: A STUDY WITH N-ETHYLMALEIMIDE AND PERTUSSIS TOXIN S. FOUCART, T.V. MURPHY AND H. MAJEWSKI 277 IMAGE 12 XVI CONTENTS PROTEIN KINASE C AND MODULATION OF NEUROTRANSMISSION: STUDIES WITH PROTEIN KINASE INHIBITORS I.F. MUSGRAVE AND H. MAJEWSKI 279 INTRASYNAPTOSOMAL PROTEIN PHOSPHORYLATION AND ITS INHIBITION BY PLASMA MEMBRANE OXIDOREDUCTASES J.-L. DREYER 281 FUNCTIONAL AND REGULATORY PROPERTIES OF PRESYNAPTIC AUTORECEPTORS OF THE 5-HTI A SUBTYPE ON DORSAL RAPHE NEURONS IN BRAIN STEM SLICES L. LANFUMEY, S. HAJ-DAHMANE, L.E. SCHECHTER, F J. BOLANOS, H. GOZLAN AND M. HAMON 285 DO SCHWANN CELLS PLAY A ROLE IN UPSTREAM REGULATION OF THE RELEASE PROBABILITY IN SYMPATHETIC NERVE VARICOSITIES? L. STJARNE, E. STJARNE, M. MSGHINA AND J.-X. BAO 289 CHANGES IN AR PRESYNAPTIC RECEPTOR SENSITIVITY DURING PRODUCTION OF DEPENDENCE TO MORPHINE IN CONSCIOUS RATS W.R. DIXON, J. MACHADO AND A.P.L. CHANG 293 ROLE OF PRESYNAPTIC 2 HETERORECEPTORS IN NONSYNAPTIC MODULATION OF TRANSMITTER RELEASE E.S. VIZI, I J. ELENKOV, F. OBERFRANK, J. KISS AND L.G. HARSING, JR. 297 AUTOREGULATION OF CATECHOLAMINE RELEASE AT CENTRAL AND SYMPATHETIC NERVE TERMINALS: COMMON FEATURES F. GONON, M.F. SUAUD-CHAGNY, C. MERMET AND L. STJARNE 303 AUTORECEPTOR MEDIATED CHANGES IN DOPAMINERGIC TERMINAL EXCITABILITY IN VIVO J. M. TEPPER 307 PREJUNCTIONAL AUTORECEPTORS IN MOUSE VAS DEFERENS K. STARKE, I. VON KIIGELGEN AND R. BIILTMANN 311 IMAGE 13 CONTENTS XVII SK & F 104078 IDENTIFIES SUBTYPES OF PREJUNCTIONAL A2-ADRENOCEPTORS IN THE RAT VAS DEFERENS R.R. RUFFOLO, JR., A J. NICHOLS, J.P. HIEBLEAND M.A. ORIOWO 315 CLONIDINE INHIBITION OF NOREPINEPHRINE RELEASE FROM NORMAL AND MORPHINE-TOLERANT GUINEA PIG CORTICAL SLICES L. BEANI, C. TOMASINI, R. GUIDORZI AND C. BIANCHI 319 HUMAN CAKI-1 CELLS ARE THE FIRST CLONAL CELL LINE KNOWN TO POSSESS THE EXTRANEURONAL TRANSPORT MECHANISM FOR NORADRENALINE (UPTAKE 2) E. SCHOMIG, C.-L. SCHONFELD AND U. TRENDELENBURG 323 INHIBITION OF NA UPTAKE BY (+)-OXAPROTIMINE INHIBITS SYMPATHETIC NERVE ACTIVITY A. SCHULTHEISS, B. SZABO AND K. STARKE 327 AUTOREGULATION OF EVOKED NORADRENALINE RELEASE AT THE SURFACE OF THE ISOLATED RAT TAIL ARTERY STUDIED BY ELECTROCHEMISTRY C. MERMET, L. STJARNE AND F. GONON 329 AUTOREGULATION OF EVOKED NORADRENALINE RELEASE IN THE RAT HYPOTHALAMIC PARAVENTRICULAR NUCLEUS STUDIED IN VIVO BY ELECTROCHEMISTRY C. MERMET, M.F. SUAUD-CHAGNY AND F. GONON 331 CLONIDINE EARLY IN LIFE: EFFECT ON BRAIN MORPHOFUNCTIONAL DISTURBANCES INDUCED BY NEONATAL MALUTRITION IN THE RAT R. SOTO-MOYANO, A. HERNANDEZ, H. PEREZ, S. RUIZ, X. GALLEGUILLOS AND J. BELMAR 333 MU AND KAPPA AGONISTS INHIBIT CARBACHOL-EVOKED RELEASE OF CATECHOLAMINES AND [MET]ENKEPHALIN FROM EX SITU PERFUSED DOG ADRENALS M.K. DOUSA, S.L. CHRITTON, C. GRABAU, T.L. YAKSH AND G.M. TYCE 335 IMAGE 14 XVIII CONTENTS ELECTROPHYSIOLOGICAL EVIDENCES FOR THE PREFERENTIAL LOCATION OF D2 AUTORECEPTORS ON DENDRITES OF DA NEURONS IN THE RAT SUBSTANTIA NIGRA P J. CHARLETY, H. AKAOKA, C.F. SAUNIER, M. BUDA AND G. CHOUVET 337 INCREASE OF POSTSYNAPTIC DOPAMINERGIC TRANSMISSION BY PRESYNAPTIC ACTIONS OF COCAINE S.P. BANERJEE, C. MANETTO AND T.I. LIDSKY 339 AUTOREGULATION OF EVOKED DOPAMINE RELEASE IN THE RAT AT CENTRAL TERMINAL SITES STUDIED IN VIVO BY ELECTROCHEMISTRY M.F. SUAUD-CHAGNY, M. BUDA AND F. GONON 341 COMBINED EFFECT OF (-)-VESAMICOL AND (+)-TUBOCURARINE ON ENDPLATE CURRENT AMPLITUDE IN RAT SKELETAL MUSCLE AT HIGH FREQUENCIES OF NERVE STIMULATION C. PRIOR, T. SEARL, K. PEMBERTON, W.C. BOWMAN AND I.G. MARSHALL 343 EFFECT OF (-)-VESAMICOL ON MINIATURE ENDPLATE CURRENT AND ENDPLATE CURRENT AMPLITUDES IN RAT SKELETAL MUSCLE T. SEARL, C. PRIOR AND I.G. MARSHALL 345 SUBJECT INDEX 347
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spellingShingle Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990
Advances in the biosciences
Récepteurs présynaptiques - Congrès
Presynaptic receptors Congresses
Receptors, Neurotransmitter drug effects Congresses
Receptors, Neurotransmitter physiology Congresses
Synaptic Transmission drug effects Congresses
Synaptic Transmission physiology Congresses
Synaptische Erregungsübertragung (DE-588)4196884-0 gnd
Rezeptor (DE-588)4049722-7 gnd
Präsynaptischer Rezeptor (DE-588)4319477-1 gnd
Synaptische Transmission (DE-588)4331218-4 gnd
Neurotransmitter-Rezeptor (DE-588)4171601-2 gnd
Präsynaptische Membran (DE-588)4315851-1 gnd
subject_GND (DE-588)4196884-0
(DE-588)4049722-7
(DE-588)4319477-1
(DE-588)4331218-4
(DE-588)4171601-2
(DE-588)4315851-1
(DE-588)1071861417
title Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990
title_auth Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990
title_exact_search Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990
title_full Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990 ed.: S. Z. Langer ...
title_fullStr Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990 ed.: S. Z. Langer ...
title_full_unstemmed Presynaptic receptors and neuronal transporters official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990 ed.: S. Z. Langer ...
title_short Presynaptic receptors and neuronal transporters
title_sort presynaptic receptors and neuronal transporters official satellite symposium to the iuphar 1990 congress held in rouen france on 26 29 june 1990
title_sub official satellite symposium to the IUPHAR 1990 congress held in Rouen, France, on 26 - 29 June 1990
topic Récepteurs présynaptiques - Congrès
Presynaptic receptors Congresses
Receptors, Neurotransmitter drug effects Congresses
Receptors, Neurotransmitter physiology Congresses
Synaptic Transmission drug effects Congresses
Synaptic Transmission physiology Congresses
Synaptische Erregungsübertragung (DE-588)4196884-0 gnd
Rezeptor (DE-588)4049722-7 gnd
Präsynaptischer Rezeptor (DE-588)4319477-1 gnd
Synaptische Transmission (DE-588)4331218-4 gnd
Neurotransmitter-Rezeptor (DE-588)4171601-2 gnd
Präsynaptische Membran (DE-588)4315851-1 gnd
topic_facet Récepteurs présynaptiques - Congrès
Presynaptic receptors Congresses
Receptors, Neurotransmitter drug effects Congresses
Receptors, Neurotransmitter physiology Congresses
Synaptic Transmission drug effects Congresses
Synaptic Transmission physiology Congresses
Synaptische Erregungsübertragung
Rezeptor
Präsynaptischer Rezeptor
Synaptische Transmission
Neurotransmitter-Rezeptor
Präsynaptische Membran
Konferenzschrift 1990 Rouen
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volume_link (DE-604)BV000003145
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