Direct Synthesis of Dihydropyrrolo[2,1‐a]Isoquinolines through FeCl3 Promoted Oxidative Aromatization

We have developed a straightforward FeCl3 promoted synthesis of dihydropyrrolo[2,1‐a]isoquinolines through formal (3+2) cycloaddition/oxidative aromatization cascade of dihydroisoquinoline with Morita‐Baylis‐Hillman carbonates (up to 96% yield). Further modifications of the obtained products were su...

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Veröffentlicht in:	Advanced synthesis & catalysis 2019-10, Vol.361 (20), p.4772-4780
Hauptverfasser:	Cui, Hai‐Lei, Jiang, Lu, Tan, Hao, Liu, Si
Format:	Artikel
Sprache:	eng
Schlagworte:	Dihydroisoquinoline Iron Chloride Morita-Baylis-Hillman carbonates Oxidative aromatization Pyrroloisoquinoline
Online-Zugang:	Volltext
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