Entry inhibitors of the HIV virus

Entry inhibitors of the HIV virus

The present invention relates to small molecules as entry inhibitors of the HIV virus, processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors...

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Hauptverfasser: Van Acker, Koenraad Lodewijk August, Wigerinck, Piet Tom Bert Paul, Michiels, Lieve Emma Jan, Tahri, Abdellah
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Sprache:eng
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creator Van Acker, Koenraad Lodewijk August
Wigerinck, Piet Tom Bert Paul
Michiels, Lieve Emma Jan
Tahri, Abdellah
description The present invention relates to small molecules as entry inhibitors of the HIV virus, processes for their preparation as well as pharmaceutical compositions, their use as medicines, and diagnostic kits comprising them. The present invention also concerns combinations of the present entry inhibitors with other anti-retroviral agents. It further relates to their use in assays as reference compounds or as reagents. The compounds of the present invention are useful for preventing or treating infection by HIV and for treating AIDS.
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title Entry inhibitors of the HIV virus
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