Process for preparing terbinafine and HCI salt thereof

Process for preparing terbinafine and HCI salt thereof

1. Field of the Invention Provided is a process for preparing terbinafine or its HCl salt comprising: reacting a furan derivative with a base to form a second compound; performing a reductive alkylation of the second compound obtained in the step with N-methyl--naphthalenemethylamine or its HCl salt...

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Hauptverfasser: Lee, Tai-Au, Wang, Kyu-Jung, Kim, Hong-Bae, Kwon, Kyoung-Chan, Ku, Chang-Hoe
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Sprache:eng
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creator Lee, Tai-Au
Wang, Kyu-Jung
Kim, Hong-Bae
Kwon, Kyoung-Chan
Ku, Chang-Hoe
description 1. Field of the Invention Provided is a process for preparing terbinafine or its HCl salt comprising: reacting a furan derivative with a base to form a second compound; performing a reductive alkylation of the second compound obtained in the step with N-methyl--naphthalenemethylamine or its HCl salt to form a third compound; and purifying the third compound.
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title Process for preparing terbinafine and HCI salt thereof
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