Novel pyrazolo[1,5-a]pyridines as PI3K inhibitors: variation of the central linker groupElectronic supplementary information (ESI) available. See DOI: 10.1039/c3md00221g

As part of our investigation into the pyrazolo[1,5- a ]pyridines as novel PI3K inhibitors, we report a range of analogues where the central linker portion of the molecule was varied while retaining the pyrazolo[1,5- a ]pyridine and arylsulfonyl or arylcarbonyl groups. Isostere generating software BR...

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Hauptverfasser:	Kendall, Jackie D, Marshall, Andrew J, Giddens, Anna C, Tsang, Kit Yee, Boyd, Maruta, Frédérick, Raphaël, Lill, Claire L, Lee, Woo-Jeong, Kolekar, Sharada, Chao, Mindy, Malik, Alisha, Yu, Shuqiao, Chaussade, Claire, Buchanan, Christina M, Rewcastle, Gordon W, Baguley, Bruce C, Flanagan, Jack U, Denny, William A, Shepherd, Peter R
Format:	Artikel
Sprache:	eng
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