Assessing Atropisomer Axial Chirality in Drug Discovery and Development
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| Veröffentlicht in: | Journal of medicinal chemistry 2011-10, Vol.54 (20), p.7005-7022 |
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| container_end_page | 7022 |
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| container_issue | 20 |
| container_start_page | 7005 |
| container_title | Journal of medicinal chemistry |
| container_volume | 54 |
| creator | LaPlante, Steven R D. Fader, Lee Fandrick, Keith R Fandrick, Daniel R Hucke, Oliver Kemper, Ray Miller, Stephen P. F Edwards, Paul J |
| description | |
| doi_str_mv | 10.1021/jm200584g |
| format | Article |
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| fulltext | fulltext |
| identifier | ISSN: 0022-2623 |
| ispartof | Journal of medicinal chemistry, 2011-10, Vol.54 (20), p.7005-7022 |
| issn | 0022-2623 1520-4804 |
| language | eng |
| recordid | cdi_proquest_miscellaneous_900630316 |
| source | MEDLINE; American Chemical Society Journals |
| subjects | Amides - chemistry Drug Discovery Heterocyclic Compounds, 4 or More Rings - chemistry Legislation, Drug Macrocyclic Compounds - chemistry Models, Molecular Pharmaceutical Preparations - chemistry Pharmacokinetics Stereoisomerism Structure-Activity Relationship Thermodynamics United States United States Food and Drug Administration |
| title | Assessing Atropisomer Axial Chirality in Drug Discovery and Development |
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