Synthesis of 4-Substituted Aminoquinoline-3-carboxylates as Potential Antimicrobial Agents
A series of 4‐substituted aminoquinoline‐3‐carboxylates was prepared and evaluated for antimicrobial activity. Four of the compounds (VIII, XIII, XV, and XXIII) exhibited low activity against Staphylococcus aureus.
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| Veröffentlicht in: | Journal of pharmaceutical sciences 1984-08, Vol.73 (8), p.1141-1143 |
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| container_end_page | 1143 |
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| container_issue | 8 |
| container_start_page | 1141 |
| container_title | Journal of pharmaceutical sciences |
| container_volume | 73 |
| creator | Mareckix, Paul E. Bambury, Ronald E. |
| description | A series of 4‐substituted aminoquinoline‐3‐carboxylates was prepared and evaluated for antimicrobial activity. Four of the compounds (VIII, XIII, XV, and XXIII) exhibited low activity against Staphylococcus aureus. |
| doi_str_mv | 10.1002/jps.2600730828 |
| format | Article |
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| fulltext | fulltext |
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| ispartof | Journal of pharmaceutical sciences, 1984-08, Vol.73 (8), p.1141-1143 |
| issn | 0022-3549 1520-6017 |
| language | eng |
| recordid | cdi_proquest_miscellaneous_81313674 |
| source | MEDLINE; Wiley Online Library All Journals; Alma/SFX Local Collection |
| subjects | 4-substituted aminoquinoline-3-carboxylates 4-Substituted aminoquinoline-3-carboxylates-synthesis 4‐Substituted aminoquinoline‐3‐carboxylates—synthesis, antimicrobial activity Aminoquinolines - chemical synthesis Aminoquinolines - pharmacology Anti-Bacterial Agents - chemical synthesis antimicrobial activity Antimicrobial agents-potential Antimicrobial agents—potential, 4‐substituted aminoquinoline‐3‐carboxylates Bacteria - drug effects Carboxylic Acids - chemical synthesis Carboxylic Acids - pharmacology Chemical Phenomena Chemistry Exact sciences and technology Heterocyclic compounds Heterocyclic compounds with only one n hetero atom and condensed derivatives Hydrolysis Microbial Sensitivity Tests Organic chemistry Preparations and properties |
| title | Synthesis of 4-Substituted Aminoquinoline-3-carboxylates as Potential Antimicrobial Agents |
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