Selective antagonists at the opiate delta-receptor

Classical opiate antagonists such as naloxone act predominantly at the opiate mu-receptor and exhibit only weak antagonism at the delta-receptor. Using two in vitro models - the field-stimulated mouse vas deferens and guinea pig ileum preparations - we have identified two novel peptide antagonists w...

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Veröffentlicht in:	Life sciences (1973) 1982-01, Vol.31 (12), p.1259-1262
Hauptverfasser:	Shaw, J.S., Miller, L., Turnbull, M.J., Gormley, J.J., Morley, J.S.
Format:	Artikel
Sprache:	eng
Schlagworte:	Analgesics, Opioid - pharmacology Animals Cyclazocine - analogs & derivatives Cyclazocine - pharmacology Enkephalin, Leucine - analogs & derivatives Enkephalin, Leucine - pharmacology Enkephalin, Methionine - pharmacology Ethylketocyclazocine Etorphine - pharmacology Guinea Pigs ileum In Vitro Techniques Male Mice Morphine Derivatives - pharmacology Narcotic Antagonists - pharmacology opiates Receptors, Opioid - drug effects Receptors, Opioid - physiology Receptors, Opioid, delta vas deferens
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