Ribose-Modified Adenosine Analogs as Potential Partial Agonists for the Adenosine Receptor

We have adopted a practical three-step route for the synthesis of 2'- and 3'-deoxy analogues of N6-substituted adenosines: protection of the hydroxyl groups, replacement of the N6-amino by a better leaving group, and combined deprotection and N6-amination in the last step. This route was u...

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