4,7 beta-Dimethyl-4-azacholestan-3-one (MK-386) and related 4-azasteroids as selective inhibitors of human type 1 5 alpha-reductase

4,7 beta-Dimethyl-4-azacholestan-3-one (MK-386) and related 4-azasteroids as selective inhibitors of human type 1 5 alpha-reductase

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Veröffentlicht in:Journal of medicinal chemistry 1994-11, Vol.37 (23), p.3871-3874
Hauptverfasser: Bakshi, R K, Patel, G F, Rasmusson, G H, Baginsky, W F, Cimis, G, Ellsworth, K, Chang, B, Bull, H, Tolman, R L, Harris, G S
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Sprache:eng
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5-alpha Reductase Inhibitors
Azasteroids - chemistry
Azasteroids - pharmacology
Humans
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container_end_page 3874
container_issue 23
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container_title Journal of medicinal chemistry
container_volume 37
creator Bakshi, R K
Patel, G F
Rasmusson, G H
Baginsky, W F
Cimis, G
Ellsworth, K
Chang, B
Bull, H
Tolman, R L
Harris, G S
description
doi_str_mv 10.1021/jm00049a003
format Article
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ispartof Journal of medicinal chemistry, 1994-11, Vol.37 (23), p.3871-3874
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source ACS Publications; MEDLINE
subjects 5-alpha Reductase Inhibitors
Azasteroids - chemistry
Azasteroids - pharmacology
Humans
title 4,7 beta-Dimethyl-4-azacholestan-3-one (MK-386) and related 4-azasteroids as selective inhibitors of human type 1 5 alpha-reductase
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