One-Pot Synthesis of Azaindoles via Palladium-Catalyzed α-Heteroarylation of Ketone Enolates

A convenient, one-pot method for the construction of a variety of azaindoles using simple ketones and haloaminopyridines is described.

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Bibliographische Detailangaben
Veröffentlicht in:	Journal of organic chemistry 2010-08, Vol.75 (15), p.5316-5319
Hauptverfasser:	Spergel, Steven H, Okoro, Danielle R, Pitts, William
Format:	Artikel
Sprache:	eng
Schlagworte:	Aza Compounds - chemical synthesis Catalysis Chemistry Exact sciences and technology Heterocyclic compounds Heterocyclic compounds with only one n hetero atom and condensed derivatives Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings Indoles - chemical synthesis Ketones - chemistry Magnetic Resonance Spectroscopy Mass Spectrometry Organic chemistry Palladium - chemistry Preparations and properties
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Beschreibung
Zusammenfassung:	A convenient, one-pot method for the construction of a variety of azaindoles using simple ketones and haloaminopyridines is described.
ISSN:	0022-3263 1520-6904
DOI:	10.1021/jo100623d