Effects of two novel non-peptide antagonists at the rabbit bradykinin B2 receptor

Large species differences have been previously observed in the pharmacology of bradykinin (BK) B2 receptor antagonists. We investigated the effect of two novel non-peptide antagonists, compound 9 (a benzodiazepine peptidomimetic related to icatibant) and the thiosemicarbazide bradyzide on the rabbit...

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Veröffentlicht in:	Peptides (New York, N.Y. : 1980) N.Y. : 1980), 2001-09, Vol.22 (9), p.1397-1402
Hauptverfasser:	Marceau, F, Houle, S, Bouthillier, J, Said, N B, Garratt, P J, Dziadulewicz, E K
Format:	Artikel
Sprache:	eng
Schlagworte:	Animals Benzodiazepinones - pharmacology Binding, Competitive - drug effects Bradykinin - analogs & derivatives Bradykinin - chemistry Bradykinin - pharmacology Bradykinin Receptor Antagonists Cells, Cultured Dose-Response Relationship, Drug Green Fluorescent Proteins Guanidines - pharmacology Humans Jugular Veins - cytology Jugular Veins - physiology Luminescent Proteins - metabolism Muscle, Smooth - drug effects Pyrrolidines - chemistry Pyrrolidines - pharmacology Rabbits Radioligand Assay Receptor, Bradykinin B2 Recombinant Fusion Proteins - pharmacokinetics Structure-Activity Relationship Thiosemicarbazones - chemistry Thiosemicarbazones - pharmacology Time Factors Tissue Distribution Transfection
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