Construction of Three Contiguous Tertiary Stereocenters from Aziridines in One Step

A range of active methylene nucleophiles were found to participate in ring-opening of tosylated aziridines under mild phase-transfer catalyzed conditions. High isolated yields coupled with a 1:1 reaction stoichiometry and high levels of relative stereocontrol are distinguishing features of this meth...

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Veröffentlicht in:	Organic letters 2007-11, Vol.9 (23), p.4677-4680
Hauptverfasser:	Blyumin, Evgeniy V, Gallon, Helen J, Yudin, Andrei K
Format:	Artikel
Sprache:	eng
Online-Zugang:	Volltext
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